SCHEMBL28755366

SCHEMBL28755366

CN(C)c1cc(=O)c2c(=O)n(C)c(=O)n(C)c2[nH]1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.62
PABPC1 P11940 1/20 0.62
GAA P10253 6/20 0.51
KMT2A Q03164 2/20 0.49
CYP2C9 P11712 2/20 0.48
CYP1A2 P05177 1/20 0.48
HTT P42858 1/20 0.46
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.37
DAO P14920 1/20 0.37
LGMN Q99538 1/20 0.37
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
DPP4 P27487 1/20 0.34
ADORA2B P29275 2/20 0.34
HSD17B10 Q99714 1/20 0.34
ADORA2A P29274 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3794609 0.69 POLB (0.56) POLBPABPC1GAAKMT2ACYP2C9
SCHEMBL3797438 0.67 POLB (0.53) POLBPABPC1GAAKMT2ACYP2C9
SCHEMBL8530149 0.62 ADORA2A (0.53) POLBPABPC1GAAKMT2ACYP1A2
SCHEMBL611080 0.60 POLB (0.45) POLBPABPC1GAAKMT2ACYP2C9
SCHEMBL2072539 0.59 ADORA2A (0.48) POLBPABPC1GAAKMT2ACYP1A2
SCHEMBL9039030 0.58 PDE3B (0.54) POLBPABPC1GAAKMT2ACYP2C9
SCHEMBL4459470 0.57 ALDH1A1 (0.63) GAAKMT2AALDH1A1PDE3BPDE3A
SCHEMBL27093179 0.56 PDE3B (0.49) POLBPABPC1CYP2C9CYP1A2KDM4E
SCHEMBL2037400 0.56 LGMN (0.66) POLBPABPC1GAAKMT2AALDH1A1
SCHEMBL20608816 0.55 LGMN (0.63) POLBPABPC1GAAKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114573582-B 1,2,3, 4-tetrahydropyrido [2,3-d ] pyrimidine compound and preparation method and application thereof 沈阳药科大学 2023-06-16 CN disclosed
CN-114573582-A 1,2,3, 4-tetrahydropyrido [2,3-d ] pyrimidine compound and preparation method and application thereof 沈阳药科大学 2022-06-03 CN disclosed