SCHEMBL3794609

SCHEMBL3794609

Cn1c(=O)c2c(=O)cn[nH]c2n(C)c1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.56
PABPC1 P11940 1/20 0.56
GAA P10253 6/20 0.46
KMT2A Q03164 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP1A2 P05177 1/20 0.43
HTT P42858 1/20 0.41
KDM4E B2RXH2 2/20 0.39
LGMN Q99538 1/20 0.37
ATAD2 Q6PL18 1/20 0.36
XDH P47989 1/20 0.36
PIK3CD O00329 2/20 0.35
ADORA3 P0DMS8 2/20 0.35
ADORA2A P29274 2/20 0.35
ADORA2B P29275 2/20 0.35
ADORA1 P30542 2/20 0.35
ALPL P05186 1/20 0.35
TMIGD3 P0DMS9 1/20 0.35
PDE4A P27815 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4430296 0.79 PDE3B (0.39) POLBPABPC1KMT2AHTTKDM4E
SCHEMBL13075951 0.73 ALDH1A1 (0.40) POLBPABPC1KMT2AHTTATAD2
SCHEMBL611080 0.72 POLB (0.45) POLBPABPC1GAAKMT2ACYP2C9
SCHEMBL28755247 0.71 POLB (1.00) POLBPABPC1GAAKMT2ACYP2C9
SCHEMBL28755504 0.71 POLB (0.66) POLBPABPC1GAAKMT2ACYP2C9
SCHEMBL28755366 0.69 POLB (0.62) POLBPABPC1GAAKMT2ACYP2C9
SCHEMBL612453 0.68 ATAD2 (0.44) GAAKMT2ACYP1A2HTTKDM4E
SCHEMBL29671977 0.66 POLB (0.57) POLBPABPC1GAAKMT2ACYP2C9
SCHEMBL11193540 0.66 PDE4A (0.44) HTTLGMNADORA2AADORA2BPDE4A
SCHEMBL28755319 0.65 POLB (0.56) POLBPABPC1GAAKMT2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125469-A1 PYRIMIDINEDIONE-FUSED HETEROCYCLIC COMPOUNDS AS TRPA1 MODULATORS GLENMARK PHARMACEUTICALS, S.A. (CH) 2010-11-04 WO disclosed