SCHEMBL28758461

SCHEMBL28758461

OCc1cc(Br)ccc1C(O)CC(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.36
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
ADRB2 P07550 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
NPC1 O15118 2/20 0.30
PDE2A O00408 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28758473 0.87 PTGDR2 (0.33) PTGDR2ADRB2
SCHEMBL29618373 0.87 PTGDR2 (0.33) PTGDR2ADRB2
SCHEMBL24517232 0.80 PTGDR2 (0.37) PTGDR2SLC6A2SLC6A4ADRB2MAPK1
SCHEMBL31394486 0.80 PTGDR2 (0.37) PTGDR2SLC6A2SLC6A4ADRB2MAPK1
SCHEMBL6673940 0.74 PTGDR2 (0.40) PTGDR2SLC6A2SLC6A4NPC1PDE2A
SCHEMBL31393937 0.74 PTGDR2 (0.40) PTGDR2SLC6A2SLC6A4NPC1PDE2A
SCHEMBL16959297 0.72 GABRA1 (0.42) PTGDR2SLC6A2SLC6A4NPC1
SCHEMBL16609146 0.70 PTGDR2 (0.40) PTGDR2SLC6A2SLC6A4MAPK1HSD17B10
SCHEMBL24517233 0.70 PTGDR2 (0.37) PTGDR2SLC6A2SLC6A4ADRB2MAPK1
SCHEMBL4100718 0.70 MAPK1 (0.41) PTGDR2ADRB2MAPK1HSD17B10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022121805-A1 FUSED RING COMPOUND AS NAV1.8 INHIBITOR AND USE THEREOF 成都康弘药业集团股份有限公司 2022-06-16 WO disclosed
CN-114591293-A Fused ring compound as Nav1.8 inhibitor and application thereof 成都康弘药业集团股份有限公司 2022-06-07 CN disclosed