SCHEMBL28778237

SCHEMBL28778237

COc1cnc2c(n1)CCCC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA3 P34903 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
MAPT P10636 1/20 0.35
CDK5 Q00535 2/20 0.33
CDK5R1 Q15078 2/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
PDGFRB P09619 2/20 0.33
PDGFRA P16234 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ACHE P22303 1/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30932863 0.82 CHRNB2 (0.42) CHRNB2CHRNA4HTR2C
SCHEMBL24638722 0.82 CHRNB2 (0.42) CHRNB2CHRNA4HTR2C
SCHEMBL18034941 0.74 MAOA (0.38) HRH3
SCHEMBL2408242 0.74 ACHE (0.38) PDGFRBPDGFRASMN1; SMN2ACHE
SCHEMBL24029391 0.73 CHRNB2 (0.34) CHRNB2CHRNA4SIRT6
SCHEMBL9014905 0.73 THRB (0.35) KMT2A
SCHEMBL9014730 0.73 CYP1A2 (0.32) HRH3
SCHEMBL4136886 0.73 NPC1 (0.48) NPC1RAB9AMAPTCDK5CDK5R1
SCHEMBL9014958 0.72 CYP1A2 (0.31) HRH3
SCHEMBL24869475 0.71 NPC1 (0.46) NPC1RAB9AMAPTCDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101454319-B Novel heterocyclic compound or salt thereof and intermediate thereof TOYAMA CHEMICAL CO LTD 2012-06-27 CN disclosed
CN-101454319-A Novel heterocyclic compound or salt thereof and intermediate thereof TOYAMA CHEMICAL CO LTD (JP) 2009-06-10 CN disclosed