SCHEMBL28784366

SCHEMBL28784366

Cc1ccc2[nH]c(-c3ccccn3)cc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 4/20 0.57
CBFB Q13951 3/20 0.55
METAP2 P50579 2/20 0.55
METAP1 P53582 2/20 0.55
NPC1 O15118 4/20 0.54
RAB9A P51151 4/20 0.54
PKM P14618 2/20 0.54
ALDH1A1 P00352 6/20 0.49
KDM4E B2RXH2 6/20 0.49
HPGD P15428 4/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
HSD17B10 Q99714 3/20 0.49
MEN1 O00255 2/20 0.49
MAPT P10636 2/20 0.49
KMT2A Q03164 2/20 0.49
LMNA P02545 2/20 0.49
GFER P55789 1/20 0.49
GSK3B P49841 2/20 0.46
CDK5 Q00535 2/20 0.46
CDK5R1 Q15078 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29470995 0.82 GSK3B (0.61) ITKMETAP2METAP1NPC1RAB9A
SCHEMBL308319 0.82 GSK3B (0.61) ITKMETAP2METAP1NPC1RAB9A
SCHEMBL1466825 0.81 SMN1; SMN2 (0.55) ITKMETAP2METAP1NPC1RAB9A
SCHEMBL6953761 0.77 KDM4E (0.54) ITKNPC1RAB9AALDH1A1KDM4E
SCHEMBL693581 0.76 GSK3B (0.59) ITKNPC1RAB9AALDH1A1KDM4E
SCHEMBL1464866 0.76 CYP19A1 (0.64) METAP1NPC1RAB9APKMALDH1A1
SCHEMBL694241 0.75 LMNA (0.49) ITKCBFBMETAP2METAP1NPC1
SCHEMBL2362656 0.75 NPC1 (0.69) ITKNPC1RAB9AALDH1A1KDM4E
SCHEMBL3005391 0.75 KDM4E (0.46) CBFBMETAP2METAP1NPC1RAB9A
SCHEMBL9669151 0.75 KDM4E (0.43) ITKCBFBMETAP2METAP1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101784543-B Indole and indazole compounds as inhibitors of cellular necrosis LG LIFE SCIENCES LTD 2013-10-16 CN disclosed
CN-101784543-A Indole and indazole compounds as inhibitors of cellular necrosis LG LIFE SCIENCES LTD 2010-07-21 CN disclosed