SCHEMBL28787353

SCHEMBL28787353

C=CC(=O)N1CCC(NC(=O)c2ccc(N)c(OC)c2)CC1

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
MCHR1 Q99705 2/20 0.46
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
AURKA O14965 1/20 0.44
AURKB Q96GD4 1/20 0.44
ACHE P22303 1/20 0.43
GPR183 P32249 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28787352 0.89 MAPKAPK2 (0.51) HTR4
SCHEMBL13575483 0.86 CRBN (0.53) HTR4ALDH1A1TSHRMCHR1KMT2A
SCHEMBL13846128 0.84 ACHE (0.49) HTR4ALDH1A1TSHRMCHR1KMT2A
SCHEMBL738237 0.84 HTR4 (0.53) HTR4MCHR1KMT2AAURKAAURKB
SCHEMBL28787322 0.83 EPHX2 (0.53) HTR4ALDH1A1TSHRMCHR1KMT2A
SCHEMBL2546256 0.83 MAPK14 (0.52) HTR4ALDH1A1KMT2AMEN1
SCHEMBL13667133 0.83 ALDH1A1 (0.45) HTR4ALDH1A1TSHRMCHR1KMT2A
SCHEMBL12894091 0.83 KMT2A (0.60) ALDH1A1TSHRMCHR1KMT2AMEN1
SCHEMBL28787314 0.83 TEAD1 (0.56) ALDH1A1KMT2AMEN1L3MBTL1
SCHEMBL13575549 0.83 KMT2A (0.46) HTR4ALDH1A1TSHRMCHR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114478539-A Novel DCLK1 inhibitor and preparation method and application thereof 中国人民解放军海军军医大学 2022-05-13 CN disclosed