SCHEMBL28790670

SCHEMBL28790670

NC=S.c1ccc2[nH]c(-n3ccnc3)nc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
HTR3A P46098 1/20 0.41
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 3/20 0.41
PKN1 Q16512 1/20 0.41
PKN2 Q16513 1/20 0.41
TP53 P04637 2/20 0.40
RAB9A P51151 3/20 0.40
MAPT P10636 2/20 0.40
CBFB Q13951 1/20 0.40
FGFR1 P11362 1/20 0.40
FLT1 P17948 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
AURKA O14965 1/20 0.40
CYP3A4 P08684 1/20 0.39
MASP2 O00187 1/20 0.39
MEN1 O00255 1/20 0.39
NUDT1 P36639 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4107024 0.91 BCHE (0.49) BCHEACHEHTR3AALDH1A1KDM4E
SCHEMBL3389271 0.77 BCHE (0.56) BCHEACHEHTR3AALDH1A1KDM4E
SCHEMBL7479170 0.71 MEN1 (0.43) MAPTCBFBCYP11B1CYP11B2CYP3A4
SCHEMBL10593475 0.71 IDO1 (0.47) TP53RAB9AAURKANPC1SMN1; SMN2
SCHEMBL15084733 0.71 NPC1 (0.39) ACHERAB9AMAPTCBFBCYP11B1
SCHEMBL1055019 0.69 CYP11B1 (0.46) KDM4ETP53RAB9AMAPTCBFB
SCHEMBL7016670 0.69 MEN1 (0.39) CBFBFGFR1FLT1CYP11B1CYP11B2
SCHEMBL11569434 0.69 AURKA (0.49) CBFBAURKACYP3A4HSD17B10ALKBH3
SCHEMBL9662962 0.67 TBXAS1 (0.52) CYP11B1CYP11B2
SCHEMBL7407358 0.66 CBFB (0.50) RAB9AMAPTCBFBFGFR1FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102066384-B Quinuclidine compounds as alpha-7 nicotinic acetylcholine receptor ligands BRISTOL MYERS SQUIBB CO 2014-07-30 CN disclosed
CN-102066384-A Quinuclidine compounds as alpha-7 nicotinic acetylcholine receptor ligands BRISTOL MYERS SQUIBB CO 2011-05-18 CN disclosed