SCHEMBL28792802

SCHEMBL28792802

O=C(O)c1sc(-c2ccc(Cl)cn2)cc1CCBr

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.35
P2RX7 Q99572 1/20 0.35
PTPN1 P18031 1/20 0.34
PTPRA P18433 1/20 0.34
ADAMTS5 Q9UNA0 1/20 0.34
BCKDK O14874 1/20 0.33
MCL1 Q07820 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
FABP4 P15090 1/20 0.33
FABP5 Q01469 1/20 0.33
KMT2A Q03164 3/20 0.33
SCD5 Q86SK9 2/20 0.33
MEN1 O00255 2/20 0.32
MAPT P10636 2/20 0.32
SCD O00767 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
SORT1 Q99523 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
COPS5 Q92905 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2170975 0.90 HDAC1 (0.36) HDAC1P2RX7PTPN1PTPRAADAMTS5
SCHEMBL2171600 0.78 NPC1 (0.40) HDAC1PTPN1PTPRAADAMTS5BCKDK
SCHEMBL2169644 0.69 PTPN1 (0.55) PTPN1PTPRAKMT2AMEN1MAPT
SCHEMBL4194300 0.68 PTPN1 (0.53) PTPN1PTPRAKMT2AMEN1MAPT
SCHEMBL2170705 0.66 GPR35 (0.32) MCL1
SCHEMBL28792719 0.66 ALDH1A1 (0.32) TSHRALDH1A1
SCHEMBL21523601 0.61 SCD5 (0.59) PTPN1SCD5MAPTSCDALDH1A1
SCHEMBL27839229 0.61 RAB9A (0.59) KMT2AMEN1MAPTLMNAL3MBTL1
SCHEMBL12344851 0.61 MEN1 (0.37) ADAMTS5FABP4FABP5KMT2ASCD5
SCHEMBL24970240 0.60 MAPT (0.40) HDAC1ADAMTS5KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102245600-A Pyrrolone melanin concentrating hormone receptor-1 antagonists BRISTOL MYERS SQUIBB CO 2011-11-16 CN disclosed