SCHEMBL28796014

SCHEMBL28796014

CC(C(=O)C(C)c1cc(N)ccc1Cl)c1cc(N)ccc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.43
TSHR P16473 2/20 0.43
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
HSD17B10 Q99714 3/20 0.39
ALDH1A1 P00352 1/20 0.39
THRB P10828 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
CASP1 P29466 1/20 0.39
RECQL P46063 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP1A2 P05177 1/20 0.39
MAPK1 P28482 1/20 0.38
ALOX5 P09917 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19862410 0.79 CYP3A4 (0.48) CYP3A4TSHRCA1CA2HSD17B10
SCHEMBL7968082 0.78 MAOA (0.39) CYP3A4TSHRCA1CA2HSD17B10
SCHEMBL1762357 0.78 CYP3A4 (0.52) CYP3A4TSHRCA1CA2HSD17B10
SCHEMBL27542431 0.78 ALDH1A1 (0.46) TSHRALDH1A1HPGDRECQLMEN1
SCHEMBL27859661 0.78 APP (0.38) ALDH1A1ALOX5
SCHEMBL28796016 0.74 CYP3A4 (0.43) CYP3A4TSHRCA1CA2HSD17B10
SCHEMBL9640869 0.74 CYP3A4 (0.52) CYP3A4TSHRCA1CA2HSD17B10
SCHEMBL27603271 0.72 CXCL8 (0.47) CYP3A4CASP1CYP1A2
SCHEMBL27859522 0.71 KDM4E (0.32) ALDH1A1KDM4ESMN1; SMN2LMNA
SCHEMBL3341272 0.71 CYP3A4 (0.44) CYP3A4TSHRHSD17B10ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102264701-A Dihydropyridone ureas as P2X7 modulators 2011-11-30 CN disclosed