SCHEMBL28796397

SCHEMBL28796397

CC(=O)c1c(C)[nH]c2c(N)cc(-c3cccnc3)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.43
AURKB Q96GD4 2/20 0.43
TTK P33981 1/20 0.43
INCENP Q9NQS7 1/20 0.43
DYRK1A Q13627 5/20 0.41
MKNK1 Q9BUB5 4/20 0.41
MKNK2 Q9HBH9 4/20 0.41
ALK Q9UM73 2/20 0.41
PIM1 P11309 2/20 0.41
CHEK1 O14757 1/20 0.41
DAPK3 O43293 1/20 0.41
JAK2 O60674 1/20 0.41
PRKD3 O94806 1/20 0.41
MAP4K4 O95819 1/20 0.41
PAK4 O96013 1/20 0.41
ABL1 P00519 1/20 0.41
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41
CSF1R P07333 1/20 0.41
RET P07949 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29635084 1.00 AURKA (0.43) AURKAAURKBTTKINCENPDYRK1A
SCHEMBL29635045 0.84 BRD4 (0.40) AURKAAURKBDYRK1AMKNK1MKNK2
SCHEMBL28796391 0.84 BRD4 (0.40) AURKAAURKBDYRK1AMKNK1MKNK2
SCHEMBL29635176 0.81 CYP11B2 (0.41) AURKAAURKBDYRK1AALKPIM1
SCHEMBL28796486 0.81 CYP11B2 (0.41) AURKAAURKBDYRK1AALKPIM1
SCHEMBL28796402 0.78 PRKCZ (0.40) AURKAAURKBDYRK1AALKPIM1
SCHEMBL29635086 0.78 ABL1 (0.50) ABL1
SCHEMBL28796403 0.78 ABL1 (0.50) ABL1
SCHEMBL29635053 0.78 PRKCZ (0.40) AURKAAURKBDYRK1AALKPIM1
SCHEMBL29635065 0.77 NAMPT (0.40) DYRK1ABRD4NR4A2TUBB4ATUBB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248472-B Anti-osteoporosis compound and derivative thereof, pharmaceutical composition, preparation method and application 中国药科大学 2022-06-28 CN claimed
CN-113248472-A Anti-osteoporosis compound and derivative thereof, pharmaceutical composition, preparation method and application 中国药科大学 2021-08-13 CN claimed
CN-113248472-B Anti-osteoporosis compound and derivative thereof, pharmaceutical composition, preparation method and application 中国药科大学 2022-06-28 CN disclosed
CN-113248472-A Anti-osteoporosis compound and derivative thereof, pharmaceutical composition, preparation method and application 中国药科大学 2021-08-13 CN disclosed