SCHEMBL29635176

SCHEMBL29635176

CC(=O)c1c(C)[nH]c2c(N3CCCC3)cc(-c3cccnc3)cc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 5/20 0.41
CYP11B1 P15538 1/20 0.41
ROCK1 Q13464 3/20 0.40
ROCK2 O75116 2/20 0.40
CDC42BPB Q9Y5S2 2/20 0.40
CDC42BPA Q5VT25 1/20 0.40
WNT1 P04628 5/20 0.40
DYRK1A Q13627 5/20 0.40
NPY5R Q15761 1/20 0.40
PIM1 P11309 2/20 0.40
BRD4 O60885 1/20 0.38
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
ALOX12 P18054 1/20 0.38
CHEK1 O14757 1/20 0.38
AURKA O14965 1/20 0.38
DAPK3 O43293 1/20 0.38
JAK2 O60674 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28796486 1.00 CYP11B2 (0.41) CYP11B2CYP11B1ROCK1ROCK2CDC42BPB
SCHEMBL28796397 0.81 AURKA (0.43) ROCK1WNT1DYRK1APIM1BRD4
SCHEMBL29635084 0.81 AURKA (0.43) ROCK1WNT1DYRK1APIM1BRD4
SCHEMBL28796391 0.79 BRD4 (0.40) ROCK1WNT1DYRK1APIM1BRD4
SCHEMBL29635045 0.79 BRD4 (0.40) ROCK1WNT1DYRK1APIM1BRD4
SCHEMBL29635053 0.76 PRKCZ (0.40) ROCK1WNT1DYRK1APIM1BRD4
SCHEMBL28362692 0.74 KDM4E (0.43) BRD4ALDH1A1ALOX12CYP3A4CYP2C9
SCHEMBL29635098 0.74 KDM4E (0.43) BRD4ALDH1A1ALOX12CYP3A4CYP2C9
SCHEMBL29635147 0.74 NPY5R (0.44) CYP11B2CYP11B1ROCK1ROCK2CDC42BPB
SCHEMBL28796393 0.74 NPY5R (0.44) CYP11B2CYP11B1ROCK1ROCK2CDC42BPB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248472-B Anti-osteoporosis compound and derivative thereof, pharmaceutical composition, preparation method and application 中国药科大学 2022-06-28 CN claimed
CN-113248472-B Anti-osteoporosis compound and derivative thereof, pharmaceutical composition, preparation method and application 中国药科大学 2022-06-28 CN disclosed