SCHEMBL28806397

SCHEMBL28806397

[c]1ccc(Nc2ccc(Cc3ccccc3)cc2)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.39
PRKAA2 P54646 1/20 0.38
CALM1 P0DP23 1/20 0.38
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
KDM4E B2RXH2 5/20 0.36
MAPT P10636 5/20 0.36
LMNA P02545 4/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 3/20 0.36
USP2 O75604 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ABCB1 P08183 2/20 0.36
ABCG2 Q9UNQ0 2/20 0.36
TDO2 P48775 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL71629 0.85 MAPT (0.47) KDM4EMAPTLMNAMEN1KMT2A
SCHEMBL988776 0.73 FABP1 (0.58) KDM4ELMNAMEN1KMT2AHPGD
SCHEMBL284700 0.73 CALM1 (0.63) CALM1ADRA2AADRA2BADRA2CMAPT
SCHEMBL10617361 0.72 CYP11B1 (0.45) CALM1IDH1
SCHEMBL19187359 0.71 ALDH1A1 (0.65) CALM1MAPTLMNAMEN1KMT2A
SCHEMBL25557237 0.71 ALDH1A1 (0.65) CALM1MAPTLMNAMEN1KMT2A
SCHEMBL4775214 0.71 NPC1 (0.53) ADRA2AKDM4EMAPTLMNAMEN1
SCHEMBL4774579 0.71 HTR7 (0.46) KDM4EMAPTLMNAMEN1KMT2A
SCHEMBL1711863 0.71 CALM1 (0.42) CALM1KDM4EMAPTLMNASMN1; SMN2
SCHEMBL13308523 0.69 ALDH1A1 (0.68) CALM1MAPTLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103201267-A AMPK-activating heterocyclic compounds and methods of use thereof RIGEL PHARMACEUTICALS INC 2013-07-10 CN claimed