SCHEMBL28808758

SCHEMBL28808758

O=S(=O)(c1cccc2[nH]ncc12)c1cccc2[nH]ncc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.54
JAK1 P23458 1/20 0.54
NOS1 P29475 4/20 0.53
AXL P30530 2/20 0.53
IDO1 P14902 3/20 0.50
METAP2 P50579 2/20 0.49
ALDH1A1 P00352 1/20 0.46
DHPS P49366 1/20 0.41
GAA P10253 1/20 0.41
HSP90AA1 P07900 1/20 0.41
CDK2 P24941 1/20 0.41
NPC1 O15118 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
BRD4 O60885 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1077138 0.85 NOS1 (0.55) JAK2JAK1NOS1AXLIDO1
SCHEMBL20789987 0.85 NOS1 (0.55) JAK2JAK1NOS1AXLIDO1
Hydrochloric Acid SCHEMBL28295355 0.84 JAK2 (0.50) JAK2JAK1NOS1AXLIDO1
SCHEMBL25468321 0.78 ALDH1A1 (0.43) JAK2JAK1NOS1AXLIDO1
SCHEMBL574814 0.75 METAP2 (0.55) JAK2JAK1NOS1AXLIDO1
SCHEMBL277054 0.74 NOS1 (0.59) JAK2JAK1NOS1AXLIDO1
SCHEMBL12601112 0.71 NOS1 (0.61) JAK2JAK1NOS1AXLIDO1
SCHEMBL29575075 0.71 NOS1 (0.55) JAK2JAK1NOS1AXLIDO1
SCHEMBL261171 0.71 NOS1 (0.55) JAK2JAK1NOS1AXLIDO1
SCHEMBL21894631 0.70 JAK2 (1.00) JAK2JAK1NOS1AXLIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103328471-A Method of making azaindazole derivatives TAKEDA PHARMACEUTICAL 2013-09-25 CN disclosed