SCHEMBL28811368

SCHEMBL28811368

Nc1cc(Oc2cncc(F)c2)ccn1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.47
NOS1 P29475 1/20 0.47
NOS2 P35228 1/20 0.47
FEN1 P39748 3/20 0.41
ALOX5AP P20292 2/20 0.41
CYP3A4 P08684 4/20 0.41
CYP1A2 P05177 3/20 0.41
CYP2C9 P11712 3/20 0.41
MET P08581 2/20 0.41
GRM5 P41594 3/20 0.38
SLC6A3 Q01959 1/20 0.37
SCN9A Q15858 1/20 0.36
MAPK14 Q16539 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29854857 1.00 NOS3 (0.47) NOS3NOS1NOS2FEN1ALOX5AP
SCHEMBL28811304 0.83 NOS3 (0.53) NOS3NOS1NOS2FEN1ALOX5AP
SCHEMBL13635718 0.80 NOS3 (0.50) NOS3NOS1NOS2FEN1ALOX5AP
SCHEMBL30635200 0.78 GRM5 (0.50) CYP3A4CYP1A2CYP2C9GRM5SLC6A3
SCHEMBL14005414 0.77 NOS3 (0.47) NOS3NOS1NOS2FEN1ALOX5AP
SCHEMBL6931821 0.77 LMNA (0.65) NOS3NOS1NOS2GRM5
SCHEMBL28810836 0.75 NOS3 (0.49) NOS3NOS1NOS2FEN1ALOX5AP
SCHEMBL4648395 0.75 NOS3 (0.52) NOS3NOS1NOS2FEN1ALOX5AP
SCHEMBL28811293 0.75 NOS3 (0.52) NOS3NOS1NOS2FEN1ALOX5AP
SCHEMBL29860750 0.75 NOS3 (0.52) NOS3NOS1NOS2FEN1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114901280-A MrgprX2 antagonists and uses thereof 德米拉公司 2022-08-12 CN disclosed