SCHEMBL13635718

SCHEMBL13635718

Nc1cc(Oc2cccc(F)c2)ccn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.50
NOS1 P29475 1/20 0.50
NOS2 P35228 1/20 0.50
FEN1 P39748 3/20 0.46
ALOX5AP P20292 2/20 0.46
MAP4K4 O95819 1/20 0.46
MET P08581 1/20 0.42
MAPK14 Q16539 1/20 0.42
KMT2A Q03164 2/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
MITF O75030 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
GFER P55789 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NLRP1 Q9C000 1/20 0.40
NOD2 Q9HC29 1/20 0.40
USP2 O75604 1/20 0.40
CDK8 P49336 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28811304 0.86 NOS3 (0.53) NOS3NOS1NOS2FEN1ALOX5AP
SCHEMBL14684302 0.82 MAOB (0.60) NOS3NOS1NOS2KMT2AMAPT
SCHEMBL24155504 0.81 DYRK1A (0.43) FEN1ALOX5APMAP4K4KMT2AMAPT
SCHEMBL30046762 0.80 NOS3 (0.55) NOS3NOS1NOS2FEN1ALOX5AP
SCHEMBL29854857 0.80 NOS3 (0.47) NOS3NOS1NOS2FEN1ALOX5AP
SCHEMBL28811368 0.80 NOS3 (0.47) NOS3NOS1NOS2FEN1ALOX5AP
SCHEMBL190964 0.79 GCK (0.51) NOS3NOS1NOS2FEN1ALOX5AP
SCHEMBL19139269 0.79 MRGPRX1 (0.45) MAP4K4MAPTALDH1A1MRGPRX1
SCHEMBL7938427 0.79 MAPT (0.46) MAP4K4KMT2AMAPTMEN1MITF
SCHEMBL11959791 0.78 LMNA (0.47) MAP4K4KMT2AMAPTMEN1MITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2119706-A1 PYRIDINE OR PYRIMIDINE DERIVATIVE HAVING EXCELLENT CELL GROWTH INHIBITION EFFECT AND EXCELLENT ANTI-TUMOR EFFECT ON CELL STRAIN HAVING AMPLIFICATION OF HGFR GENE Eisai R&D Management Co., Ltd. (JP) 2009-11-18 EP disclosed