SCHEMBL28811657

SCHEMBL28811657

FC(F)(F)c1cccc(Nc2cnc3ccccc3c2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH2 P48735 2/20 0.56
KIF11 P52732 1/20 0.55
ABCG2 Q9UNQ0 3/20 0.54
EGFR P00533 1/20 0.54
TSHR P16473 1/20 0.53
HTT P42858 1/20 0.53
MTOR P42345 1/20 0.53
IGF1R P08069 2/20 0.52
AURKA O14965 2/20 0.50
CTSC P53634 1/20 0.50
TRPV1 Q8NER1 1/20 0.50
ALPL P05186 1/20 0.49
KDM4E B2RXH2 1/20 0.49
ULK1 O75385 1/20 0.48
SLC22A12 Q96S37 1/20 0.48
ALDH1A1 P00352 1/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29801795 1.00 IDH2 (0.56) IDH2KIF11ABCG2EGFRTSHR
SCHEMBL2111139 0.80 KDM4E (0.58) HTTIGF1RKDM4EALDH1A1MAPT
SCHEMBL1702912 0.79 IGF1R (0.48) IGF1RTRPV1ALPLULK1SLC22A12
SCHEMBL18796092 0.79 ALPL (0.48) IGF1RTRPV1ALPLULK1SLC22A12
SCHEMBL878873 0.78 CDK8 (0.59) IDH2KIF11AURKACTSCKDM4E
SCHEMBL7697641 0.78 AURKA (0.54) IDH2KIF11ABCG2EGFRTSHR
SCHEMBL17742433 0.78 IGF1R (0.51) ABCG2IGF1RKDM4ERAB9ASMN1; SMN2
SCHEMBL3952943 0.78 IGF1R (0.72) ABCG2EGFRIGF1RALPLKDM4E
SCHEMBL394991 0.78 KIF11 (0.70) IDH2KIF11HTTAURKAKDM4E
SCHEMBL23553607 0.77 VCP (0.64) ABCG2MTORKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114736156-A Preparation method and application of simplified derivatives of cryptolepine 中捷四方生物科技股份有限公司 2022-07-12 CN disclosed