SCHEMBL28813152

SCHEMBL28813152

O=[N+]([O-])c1ccc(CNc2ccc3ncoc3c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPRF P10586 1/20 0.51
PTPN2 P17706 1/20 0.51
PTPN1 P18031 1/20 0.51
PTPN11 Q06124 1/20 0.51
MAPT P10636 4/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
PSEN1 P49768 1/20 0.44
PSEN2 P49810 1/20 0.44
APH1B Q8WW43 1/20 0.44
NCSTN Q92542 1/20 0.44
APH1A Q96BI3 1/20 0.44
PSENEN Q9NZ42 1/20 0.44
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7029620 0.78 CYP3A4 (0.49) PTPN1MAPTMEN1KMT2AALDH1A1
SCHEMBL2542456 0.76 CYP3A4 (0.61) PTPRFPTPN2PTPN1PTPN11MAPT
SCHEMBL4953680 0.76 PTPRF (0.83) PTPRFPTPN2PTPN1PTPN11MAPT
SCHEMBL27971027 0.75 PTPRF (0.51) PTPRFPTPN2PTPN1PTPN11MAPT
SCHEMBL27971024 0.75 LMNA (0.45) PTPN1PTPN11MAPTMEN1KMT2A
SCHEMBL6699468 0.73 PTPRF (0.78) PTPRFPTPN2PTPN1PTPN11MAPT
SCHEMBL27970900 0.73 LMNA (0.43) PTPN1PTPN11MAPTMEN1KMT2A
SCHEMBL22783774 0.72 PTPRF (0.75) PTPRFPTPN2PTPN1PTPN11MAPT
SCHEMBL10938044 0.72 PTPRF (0.60) PTPRFPTPN2PTPN1PTPN11MAPT
SCHEMBL531299 0.72 PTPRF (0.60) PTPRFPTPN2PTPN1PTPN11MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103992310-A Group of substituted benzoheterocycle amine derivatives and preparation method and related application thereof as IMPDH (inosine monophosphate dehydrogenase) inhibitor INST MEDICINAL BIOTECHNOLOGY 2014-08-20 CN disclosed