SCHEMBL28816481

SCHEMBL28816481

COP(=O)(CC(=O)[C@H](CC1CN(OC(=O)C(C)(C)C)C1)NC(=O)OCc1ccccc1)OC

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KYNU Q16719 1/20 0.44
CTSL P07711 6/20 0.40
CTSK P43235 5/20 0.40
CTSS P25774 4/20 0.40
CTSB P07858 2/20 0.40
BCHE P06276 2/20 0.40
ACHE P22303 2/20 0.40
CACNA1F O60840 1/20 0.40
CACNA1D Q01668 1/20 0.40
CACNA1S Q13698 1/20 0.40
CACNA1C Q13936 1/20 0.40
CASP1 P29466 4/20 0.40
ALDH1A1 P00352 1/20 0.39
ALOX15 P16050 1/20 0.39
SYK P43405 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27835434 1.00 KYNU (0.44) KYNUCTSLCTSKCTSSCTSB
SCHEMBL28816503 0.92 CTSK (0.42) KYNUCTSLCTSKCTSSCTSB
SCHEMBL27998434 0.89 BCHE (0.44) KYNUCTSLCTSKCTSSCTSB
SCHEMBL478953 0.86 KYNU (0.44) KYNUCTSLCTSKCTSSSYK
SCHEMBL478951 0.86 KYNU (0.44) KYNUCTSLCTSKCTSSSYK
SCHEMBL3410144 0.81 KYNU (0.50) KYNUCTSLCTSKCTSSCTSB
SCHEMBL478461 0.80 ACKR3 (0.46) CTSLCTSKCTSSCTSBBCHE
SCHEMBL478463 0.80 ACKR3 (0.46) CTSLCTSKCTSSCTSBBCHE
Tert-Butyl Formate SCHEMBL27835436 0.78 KYNU (0.43) KYNUCTSLCTSKCTSSCTSB
SCHEMBL478742 0.78 YAP1 (0.45) CTSLBCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102026996-B Pyridazine derivatives as factor XIA inhibitors BRISTOL MYERS SQUIBB CO 2015-01-07 CN disclosed