SCHEMBL3410144

SCHEMBL3410144

COP(=O)(CC(=O)C(CC1CNC1)NC(=O)OCc1ccccc1)OC

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KYNU Q16719 1/20 0.50
CTSK P43235 6/20 0.45
CTSL P07711 5/20 0.45
CTSS P25774 4/20 0.45
CTSB P07858 4/20 0.45
CASP1 P29466 3/20 0.44
ALDH1A1 P00352 1/20 0.43
ALOX15 P16050 1/20 0.43
TACR1 P25103 1/20 0.43
IDO1 P14902 2/20 0.42
TDO2 P48775 1/20 0.42
ELANE P08246 1/20 0.42
PRTN3 P24158 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tert-Butyl Formate SCHEMBL27835436 0.92 KYNU (0.43) KYNUCTSKCTSLCTSSCTSB
Tert-Butyl Formate SCHEMBL28816504 0.84 CTSL (0.42) KYNUCTSKCTSLCTSSCTSB
SCHEMBL28816481 0.81 KYNU (0.44) KYNUCTSKCTSLCTSSCTSB
SCHEMBL478951 0.81 KYNU (0.44) KYNUCTSKCTSLCTSS
SCHEMBL27835434 0.81 KYNU (0.44) KYNUCTSKCTSLCTSSCTSB
SCHEMBL480359 0.78 SYK (0.61) KYNUCTSKCTSLCTSSCTSB
Tert-Butyl Formate SCHEMBL27998436 0.78 ITGB3 (0.50) KYNUCTSKCTSLCTSBCASP1
SCHEMBL478463 0.77 ACKR3 (0.46) CTSKCTSLCTSSCTSB
SCHEMBL478461 0.77 ACKR3 (0.46) CTSKCTSLCTSSCTSB
SCHEMBL28816503 0.77 CTSK (0.42) KYNUCTSKCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2265601-A1 PYRIDAZINE DERIVATIVES AS FACTOR XIA INHIBITORS Bristol-Myers Squibb Company (US) 2010-12-29 EP disclosed
WO-2009114677-A1 PYRIDAZINE DERIVATIVES AS FACTOR XIA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-09-17 WO disclosed