SCHEMBL28817124

SCHEMBL28817124

CC(COC(N)=O)c1ccc(B2OC(C)(C)C(C)(C)O2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.45
F11 P03951 4/20 0.45
CA1 P00915 4/20 0.43
CA2 P00918 4/20 0.43
CA9 Q16790 4/20 0.43
F2 P00734 3/20 0.42
PRSS1 P07477 2/20 0.42
PRSS2 P07478 2/20 0.42
PRSS3 P35030 2/20 0.42
LIPG Q9Y5X9 8/20 0.40
LPL P06858 7/20 0.40
CA12 O43570 1/20 0.40
CA3 P07451 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
CA5A P35218 1/20 0.40
CA7 P43166 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CA5B Q9Y2D0 1/20 0.40
AAK1 Q2M2I8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28817123 1.00 ESR2 (0.45) ESR2F11CA1CA2CA9
SCHEMBL28817201 0.85 CYP1A2 (0.40) ESR2F11CA1CA2CA9
SCHEMBL28817105 0.81 AAK1 (0.47) ESR2F11CA1CA2CA9
SCHEMBL28817172 0.81 CYP1A2 (0.34) ESR2F11CA1CA2CA9
SCHEMBL28623122 0.79 CA1 (0.46) ESR2F11CA1CA2CA9
SCHEMBL28623123 0.79 CA1 (0.46) ESR2F11CA1CA2CA9
SCHEMBL21472005 0.79 P4HB (0.39) ESR2F11CA1CA2CA9
SCHEMBL17129624 0.78 DGAT1 (0.44) ESR2F11CA1CA2CA9
SCHEMBL15778480 0.77 LIPG (0.42) ESR2F11CA1CA2CA9
SCHEMBL5336869 0.77 F11 (0.56) ESR2F11CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108341774-B Substituted quinolinone inhibitors 首药控股(北京)股份有限公司 2022-07-19 CN disclosed