SCHEMBL28819009

SCHEMBL28819009

NC(=O)c1nc(-c2ccccc2)c([N+](=O)[O-])s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.45
KMT2A Q03164 6/20 0.45
MEN1 O00255 5/20 0.45
MAPT P10636 2/20 0.45
HTT P42858 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
PKM P14618 1/20 0.45
MAPK1 P28482 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CDC7 O00311 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
DBF4 Q9UBU7 1/20 0.43
KDM4E B2RXH2 3/20 0.40
CYP1A2 P05177 1/20 0.39
POLB P06746 3/20 0.38
GAA P10253 2/20 0.38
SCN9A Q15858 1/20 0.38
PTGS2 P35354 1/20 0.38
LIMK1 P53667 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11040221 0.78 ALDH1A1 (0.64) ALDH1A1KMT2AMEN1MAPTHTT
SCHEMBL12127937 0.78 ALDH1A1 (0.56) ALDH1A1KMT2AMEN1MAPTHTT
SCHEMBL27757739 0.76 CDC7 (0.55) ALDH1A1KMT2AMEN1MAPTHTT
SCHEMBL3308450 0.76 SCN9A (0.57) ALDH1A1KMT2AMEN1MAPTSMN1; SMN2
SCHEMBL11456650 0.76 PTGDR2 (0.49) ALDH1A1KMT2AMEN1MAPTHTT
SCHEMBL3456228 0.73 ADORA2B (0.62) ALDH1A1MAPTHTTSMN1; SMN2NPSR1
SCHEMBL3311788 0.73 ALDH1A1 (0.60) ALDH1A1MAPTSMN1; SMN2KDM4ECYP1A2
SCHEMBL28017851 0.73 ALDH1A1 (0.52) ALDH1A1CDC7CCNE1CDK2DBF4
SCHEMBL25063308 0.72 KMT2A (0.56) ALDH1A1KMT2AMEN1MAPTSMN1; SMN2
SCHEMBL3168556 0.72 DGAT1 (0.53) ALDH1A1KMT2AMEN1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104592152-A Amidine structure containing nitrobenzene thiazolecarboxylic acid amide dual-target inhibitor, as well as preparation method and application thereof FOSHAN SAIWEISI PHARMACEUTICAL TECHNOLOGY CO LTD 2015-05-06 CN disclosed