SCHEMBL28819092

SCHEMBL28819092

CS(=O)(=O)Nc1ccc(NC(=O)c2ccc(F)cc2C(F)(F)F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR27 Q9NS67 4/20 0.54
AVPR2 P30518 3/20 0.54
KIF11 P52732 2/20 0.50
TRPV1 Q8NER1 1/20 0.48
NR3C2 P08235 2/20 0.48
AURKA O14965 4/20 0.48
CHEK2 O96017 1/20 0.48
CSF1R P07333 1/20 0.48
RET P07949 1/20 0.48
FLT4 P35916 1/20 0.48
ABL2 P42684 1/20 0.48
BLK P51451 1/20 0.48
LIMK1 P53667 1/20 0.48
AURKB Q96GD4 1/20 0.48
TRPV4 Q9HBA0 1/20 0.45
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL679036 0.81 PTGS1 (0.52) GPR27AVPR2TRPV1AURKACHEK2
SCHEMBL23002357 0.79 GPR27 (0.48) GPR27AVPR2NR3C2KDM4ELMNA
SCHEMBL12334377 0.78 RORC (0.58) GPR27AVPR2TRPV1AURKACHEK2
SCHEMBL31240769 0.76 KIF11 (0.51) GPR27AVPR2KIF11MEN1KMT2A
SCHEMBL1160927 0.75 HDAC1 (0.52) TRPV1AURKACHEK2CSF1RRET
SCHEMBL1417617 0.74 KMT2A (0.49) AURKACHEK2CSF1RRETFLT4
SCHEMBL7319545 0.73 ORAI1 (0.66) AURKACHEK2CSF1RRETFLT4
SCHEMBL13485802 0.73 LMNA (0.61) AURKACHEK2CSF1RRETFLT4
SCHEMBL27801156 0.72 AURKA (0.49) GPR27AVPR2NR3C2AURKACHEK2
SCHEMBL30133947 0.72 KMT2A (0.49) KIF11AURKACHEK2CSF1RRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102573994-B Novel bicyclic urea compounds MERCK PATENT GMBH 2015-06-24 CN disclosed