SCHEMBL28820131

SCHEMBL28820131

COc1ccnc(OCc2ccncc2)n1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LOX P28300 1/20 0.41
LOXL2 Q9Y4K0 1/20 0.41
ABCB1 P08183 2/20 0.40
RXRA P19793 5/20 0.40
GRIN1 Q05586 5/20 0.40
GRIN2B Q13224 5/20 0.40
PIK3CA P42336 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CYP17A1 P05093 1/20 0.38
PLK1 P53350 1/20 0.37
IKBKB O14920 1/20 0.37
PIK3C3 Q8NEB9 1/20 0.36
MGMT P16455 1/20 0.36
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28619751 0.87 ALDH1A1 (0.50) RXRAGRIN1GRIN2BALDH1A1
SCHEMBL12015 0.76 CCR1 (0.41) LOXLOXL2RXRAGRIN1GRIN2B
SCHEMBL29520064 0.76 CCR1 (0.41) LOXLOXL2RXRAGRIN1GRIN2B
SCHEMBL27990718 0.74 CCR1 (0.40) LOXLOXL2RXRAGRIN1GRIN2B
SCHEMBL4271456 0.74 ALKBH1 (0.47) ALDH1A1
SCHEMBL28020288 0.74 MAPK8 (0.42) LOXLOXL2RXRAGRIN1GRIN2B
SCHEMBL28020330 0.74 TSHR (0.38) LOXLOXL2RXRAGRIN1GRIN2B
SCHEMBL16815519 0.73 RXRA (0.43) ABCB1RXRAGRIN1GRIN2BPIK3CA
SCHEMBL30721403 0.72 LOX (0.40) LOXLOXL2RXRAGRIN1GRIN2B
SCHEMBL8670180 0.72 AOC3 (0.41) PIK3CAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104725397-A Thienopyrimidine derivatives, a process for their preparation and pharmaceutical compositions containing them SERVIER LAB 2015-06-24 CN disclosed