SCHEMBL28820148

SCHEMBL28820148

CC(C)(C)C(=O)On1ncc2cc(C#C[Si](C)(C)C)ccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 8/20 0.38
GABRA1 P14867 7/20 0.38
GABRG2 P18507 6/20 0.38
GABRB3 P28472 6/20 0.38
GABRA3 P34903 5/20 0.38
GABRA2 P47869 5/20 0.38
GABRA6 Q16445 4/20 0.38
HAO1 Q9UJM8 2/20 0.35
GABRA4 P48169 5/20 0.33
CYP11B2 P19099 1/20 0.33
GABRB2 P47870 1/20 0.33
SMO Q99835 1/20 0.32
CHEK1 O14757 1/20 0.31
AURKA O14965 1/20 0.31
DAPK3 O43293 1/20 0.31
CSNK1A1 P48729 1/20 0.31
GSK3A P49840 1/20 0.31
LIMK1 P53667 1/20 0.31
IKBKE Q14164 1/20 0.31
MAPK14 Q16539 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27810079 0.78 GABRA5 (0.42) GABRA5GABRA1GABRG2GABRB3GABRA3
SCHEMBL27634812 0.77 CHEK1 (0.54) CYP11B2SMOCHEK1AURKADAPK3
SCHEMBL27690302 0.77 HDAC8 (0.39) SMOCHEK1AURKADAPK3CSNK1A1
SCHEMBL4014826 0.75 CHEK1 (0.57) GABRA5GABRA1GABRG2GABRB3GABRA3
SCHEMBL4293893 0.75 CHEK1 (0.43) GABRA5GABRA1GABRG2GABRB3GABRA3
SCHEMBL27664784 0.74 KMO (0.41) CYP11B2
SCHEMBL27634814 0.73 GLS (0.47) CLK4
SCHEMBL28001357 0.73 NOTUM (0.33) CYP11B2SMOCHEK1AURKADAPK3
SCHEMBL28995765 0.72 GRIN2B (0.46) HAO1
SCHEMBL27769204 0.71 CHEK1 (0.32) SMOCHEK1AURKADAPK3CSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103429585-B Indazolyl triazole derivatives as interleukin-1 receptor associated kinase inhibitors MERCK SERONO SA 2015-07-08 CN disclosed