SCHEMBL28823672

SCHEMBL28823672

COc1ccc2c(c1)CCCNC2C=O

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.49
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47
CA14 Q9ULX7 2/20 0.47
CA7 P43166 1/20 0.47
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
CHRNA7 P36544 1/20 0.42
DRD1 P21728 1/20 0.41
SRD5A1 P18405 2/20 0.40
HTR2A P28223 1/20 0.40
HTR2B P41595 1/20 0.40
KDM1A O60341 1/20 0.40
CYP19A1 P11511 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17732726 0.91 CA1 (0.55) HTR2CCA1CA2CA9CA14
SCHEMBL17732708 0.91 CA1 (0.55) HTR2CCA1CA2CA9CA14
SCHEMBL17732716 0.91 CA1 (0.55) HTR2CCA1CA2CA9CA14
SCHEMBL28823734 0.85 CA1 (0.50) CA1CA2CA9CA14CA7
SCHEMBL28823799 0.82 PPARD (0.41) HTR2C
SCHEMBL28823708 0.79 CAMK2A (0.47) HTR2CKMT2AMEN1SRD5A1HTR2A
SCHEMBL28823682 0.79 HTR2C (0.43) HTR2CSRD5A1HTR2AHTR2BKDM1A
SCHEMBL28823725 0.78 LRRK2 (0.42) KDM1ACYP19A1
SCHEMBL28967711 0.75 PRCP (0.42)
SCHEMBL19453963 0.75 CA1 (0.60) HTR2CCA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114929691-A Bicyclic compounds and uses thereof 爱思开生物制药株式会社 2022-08-19 CN disclosed