SCHEMBL28825121

SCHEMBL28825121

COc1cc(-c2nnc(S)n2N)c([N+](=O)[O-])c(OC)c1OC

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.45
ALDH1A1 P00352 4/20 0.37
HTT P42858 1/20 0.36
MCL1 Q07820 1/20 0.35
SOST Q9BQB4 1/20 0.35
LMNA P02545 2/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 2/20 0.34
TSHR P16473 1/20 0.34
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
CTDSP1 Q9GZU7 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GAA P10253 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28279054 0.74 KDM4E (0.41) ALDH1A1HTTLMNATSHRKDM4E
SCHEMBL2895238 0.74 ALDH1A1 (0.53) ALDH1A1HTTLMNAKMT2ATSHR
SCHEMBL28046895 0.72 PKM (0.50) PKMALDH1A1HTTMCL1LMNA
SCHEMBL9348700 0.70 PKM (0.65) PKMALDH1A1HTTMCL1LMNA
SCHEMBL4483317 0.69 ALDH1A1 (0.42) ALDH1A1LMNAKMT2ATSHRKDM4E
SCHEMBL4486268 0.69 ACHE (0.42) ALDH1A1LMNAKMT2ATSHRKDM4E
SCHEMBL2905398 0.69 PKM (0.59) PKMALDH1A1HTTMCL1LMNA
SCHEMBL2893131 0.69 ALDH1A1 (0.45) ALDH1A1LMNAKMT2ATSHRKDM4E
SCHEMBL2889816 0.68 KDM4E (0.52) ALDH1A1LMNAKMT2ATSHRKDM4E
SCHEMBL4351022 0.68 MEN1 (0.47) ALDH1A1LMNAKMT2ATDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105330651-A 1,2,4-Triazolethione derivative containing (hetero)aryl group and piperazine, and preparation method and application thereof UNIV NANKAI 2016-02-17 CN disclosed