SCHEMBL4723906

SCHEMBL4723906

Nc1ccccc1-n1nc(-c2cccc(C(F)(F)F)c2)ccc1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.51
XDH P47989 1/20 0.46
ALDH1A1 P00352 3/20 0.44
HPGD P15428 2/20 0.44
KDM4E B2RXH2 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
GABRA1 P14867 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA2 P47869 1/20 0.44
HSD17B10 Q99714 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
LMNA P02545 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MAOB P27338 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4721881 0.81 GAA (0.43) HDAC1ALDH1A1HPGDKDM4ECYP1A2
SCHEMBL4723245 0.81 KDM4E (0.51) HDAC1KDM4ETDP1LMNANPSR1
SCHEMBL14973530 0.74 ALDH1A1 (0.50) HDAC1ALDH1A1HPGDKDM4ECYP1A2
SCHEMBL22633138 0.69 TLR8 (0.51) XDHALDH1A1HPGDKDM4ECYP1A2
SCHEMBL9383785 0.68 KDM4E (0.56) XDHALDH1A1HPGDKDM4ECYP1A2
SCHEMBL13733242 0.68 ALDH1A1 (0.52) XDHALDH1A1HPGDKDM4ECYP1A2
SCHEMBL28825532 0.68 CYP1A2 (0.49) ALDH1A1HPGDKDM4ECYP1A2CYP3A4
SCHEMBL6697417 0.67 ALDH1A1 (0.66) ALDH1A1HPGDKDM4ECYP1A2CYP3A4
SCHEMBL1032856 0.67 KDM1A (0.50) XDHALDH1A1HPGDKDM4ECYP1A2
SCHEMBL27409555 0.67 HDAC1 (0.49) HDAC1XDHALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP claimed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed