SCHEMBL28825609

SCHEMBL28825609

COc1ncccc1[CH]c1ccc(F)c(C(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 7/20 0.42
GRIN2B Q13224 7/20 0.42
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
IDH1 O75874 1/20 0.34
NFE2L2 Q16236 5/20 0.33
RXRA P19793 5/20 0.33
SOS1 Q07889 2/20 0.32
APLNR P35414 1/20 0.32
RELA Q04206 1/20 0.32
FFAR4 Q5NUL3 1/20 0.31
CTSA P10619 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825671 0.84 GRIN1 (0.45) GRIN1GRIN2BALOX5APFEN1NFE2L2
SCHEMBL28825503 0.72 MEN1 (0.41) GRIN1GRIN2BNFE2L2RXRA
SCHEMBL12094716 0.71 APLNR (0.43) GRIN1GRIN2BALOX5APFEN1SOS1
SCHEMBL30864870 0.71 APLNR (0.43) GRIN1GRIN2BALOX5APFEN1SOS1
SCHEMBL28825599 0.71 GRIN1 (0.46) GRIN1GRIN2BIDH1RXRA
SCHEMBL28825611 0.71 GRIN1 (0.43) GRIN1GRIN2BRXRA
SCHEMBL28825666 0.69 GRIN1 (0.41) GRIN1GRIN2BRXRARELA
SCHEMBL28825504 0.69 ALOX5 (0.42) GRIN1GRIN2BNFE2L2
SCHEMBL23516654 0.68 IDH1 (0.44) IDH1NFE2L2APLNR
SCHEMBL28151579 0.68 IDH1 (0.44) ALOX5APFEN1IDH1NFE2L2APLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed