SCHEMBL28825638

SCHEMBL28825638

Cc1cncc([CH]c2ccc(F)c(F)c2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 2/20 0.49
CYP11B1 P15538 3/20 0.37
CYP11B2 P19099 3/20 0.37
TRPA1 O75762 1/20 0.36
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP1B1 Q16678 1/20 0.35
GRIN1 Q05586 2/20 0.34
GRIN2B Q13224 2/20 0.34
KDM1A O60341 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
NTSR1 P30989 1/20 0.33
PLA2G7 Q13093 2/20 0.33
PABPC1 P11940 1/20 0.33
RAB9A P51151 1/20 0.33
EIF4H Q15056 1/20 0.33
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
PLEC Q15149 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28825624 0.84 GRIN2B (0.39) NFE2L2CYP11B1CYP11B2GRIN1GRIN2B
SCHEMBL28825579 0.82 NFE2L2 (0.46) NFE2L2CYP11B1CYP11B2TRPA1CYP1A1
SCHEMBL28825598 0.82 GRIN2B (0.41) NFE2L2CYP11B1CYP11B2GRIN1GRIN2B
SCHEMBL28825625 0.79 GRIN1 (0.43) GRIN1GRIN2B
SCHEMBL28825596 0.79 ROCK2 (0.50) NFE2L2CYP11B1CYP11B2CYP1A1CYP1A2
SCHEMBL28523455 0.78 NFE2L2 (0.41) NFE2L2CYP11B1CYP11B2TRPA1CYP1A1
SCHEMBL28825475 0.77 CYP1A1 (0.52) NFE2L2CYP11B1CYP11B2CYP1A1CYP1A2
SCHEMBL3299908 0.77 NFE2L2 (0.54) NFE2L2TRPA1CYP1A1CYP1A2CYP1B1
SCHEMBL28825627 0.73 KCNQ3 (0.41) NFE2L2TRPA1CYP1A1CYP1A2CYP1B1
SCHEMBL8485821 0.68 VCP (0.41) CYP11B1CYP11B2RAB9ACYP2A6HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed