SCHEMBL28825596

SCHEMBL28825596

COc1cncc([CH]c2ccc(F)c(F)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.50
MAP4K4 O95819 1/20 0.50
PRKACA P17612 1/20 0.50
ROCK1 Q13464 1/20 0.50
DYRK1A Q13627 1/20 0.50
NTRK3 Q16288 1/20 0.50
PKN2 Q16513 1/20 0.50
CLK4 Q9HAZ1 1/20 0.50
MKNK2 Q9HBH9 1/20 0.50
STK17A Q9UEE5 1/20 0.50
CYP11B1 P15538 5/20 0.40
CYP11B2 P19099 4/20 0.40
NQO2 P16083 2/20 0.39
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
NFE2L2 Q16236 3/20 0.38
MAPT P10636 1/20 0.38
CYP1A2 P05177 4/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28696701 0.85 ROCK2 (0.46) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL28949613 0.84 CYP11B2 (0.51) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL28825637 0.84 NQO2 (0.53) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL28825560 0.83 CYP11B1 (0.44) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL28825677 0.82 GRIN1 (0.45) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL28825638 0.79 NFE2L2 (0.49) CYP11B1CYP11B2GRIN1GRIN2BNFE2L2
SCHEMBL28825579 0.78 NFE2L2 (0.46) CYP11B1CYP11B2GRIN1GRIN2BNFE2L2
SCHEMBL28825675 0.78 ROCK2 (0.50) ROCK2MAP4K4PRKACAROCK1DYRK1A
SCHEMBL28523455 0.74 NFE2L2 (0.41) CYP11B1CYP11B2NFE2L2MAPTCYP1A2
SCHEMBL3299908 0.73 NFE2L2 (0.54) GRIN1GRIN2BNFE2L2MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114007610-A Substituted heteroaromatic pyrazolopyridines and their use as modulators of the GLUN2B receptor 詹森药业有限公司 2022-02-01 CN disclosed