SCHEMBL28825720

SCHEMBL28825720

CC(=O)Oc1c(O)c2cc(NC(=O)c3ccccc3)ccc2n(C)c1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.53
NGFR P08138 1/20 0.53
MAPT P10636 2/20 0.48
POLB P06746 1/20 0.48
EGFR P00533 2/20 0.47
SRC P12931 2/20 0.47
TP53 P04637 1/20 0.46
NPC1 O15118 3/20 0.44
KMT2A Q03164 2/20 0.44
RAB9A P51151 2/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
TOP1 P11387 2/20 0.44
BRPF1 P55201 2/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
RECQL P46063 1/20 0.43
ALOX15 P16050 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28049574 0.84 GAA (0.52) MAPTNPC1KMT2ARAB9AMEN1
SCHEMBL28211409 0.82 NTRK1 (0.56) NTRK1NGFRMAPTPOLBEGFR
SCHEMBL19086870 0.81 NPC1 (0.53) NTRK1NGFRMAPTPOLBEGFR
SCHEMBL7975873 0.80 MAPT (0.52) NTRK1NGFRMAPTPOLBEGFR
SCHEMBL28211430 0.80 NTRK1 (0.54) NTRK1NGFRMAPTPOLBEGFR
SCHEMBL6581634 0.78 ALDH1A1 (0.54) MAPTTP53NPC1RAB9AALDH1A1
SCHEMBL6578990 0.77 ALDH1A1 (0.64) NPC1KMT2ARAB9AMEN1ALDH1A1
SCHEMBL17578567 0.77 HIF1A (0.67) NPC1KMT2ARAB9AMEN1
SCHEMBL7998977 0.76 TP53 (0.46) NTRK1NGFRMAPTPOLBSRC
SCHEMBL7997564 0.75 TP53 (0.50) MAPTPOLBTP53NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384687-A Quinolinone compound and application thereof in drugs GUANGDONG HEC PHARMACEUTICAL 2016-03-09 CN disclosed