SCHEMBL28826421

SCHEMBL28826421

COc1ccc(CC2(N)C=C(N)C=CN2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.38
AGXT P21549 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38
SLC6A4 P31645 1/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 2/20 0.35
MAPK1 P28482 1/20 0.35
ALDH1A1 P00352 3/20 0.35
MAOB P27338 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
ALOX15 P16050 1/20 0.35
CYP2D6 P10635 2/20 0.35
ATM Q13315 1/20 0.35
MMP2 P08253 2/20 0.35
MMP9 P14780 2/20 0.35
MMP8 P22894 2/20 0.35
MMP13 P45452 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4456076 0.73 ALDH1A1 (0.38) IDO1AGXTTAAR1SLC6A4POLB
SCHEMBL25227714 0.67 SMN1; SMN2 (0.43) MEN1KMT2AMAPK1ALDH1A1KDM4E
SCHEMBL1824702 0.65 MAOB (0.55) IDO1AGXTTAAR1SLC6A4ALDH1A1
Hydrochloric Acid SCHEMBL30293103 0.64 MAOB (0.53) IDO1AGXTTAAR1SLC6A4TDP1
SCHEMBL9602890 0.64 ALDH1A1 (0.37) IDO1AGXTTAAR1SLC6A4POLB
SCHEMBL1822033 0.63 MAOB (0.47) IDO1AGXTTAAR1SLC6A4MAOB
SCHEMBL491284 0.63 IDO1 (0.42) IDO1AGXTTAAR1SLC6A4ALDH1A1
SCHEMBL4868046 0.62 TDP1 (0.52) IDO1AGXTTAAR1SLC6A4POLB
Hydrochloric Acid SCHEMBL3966019 0.62 IDO1 (0.47) IDO1AGXTTAAR1SLC6A4MAOB
SCHEMBL1824988 0.62 SLC6A4 (0.46) IDO1AGXTTAAR1SLC6A4MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102770426-B As compound and the composition of kinases inhibitor NOVARTIS AG (CH) 2016-03-23 CN disclosed