SCHEMBL4456076

SCHEMBL4456076

COc1ccc(CC2(N)N=C(N)C=CN2)cc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
CYP2D6 P10635 1/20 0.38
ATM Q13315 1/20 0.38
IDO1 P14902 3/20 0.38
AGXT P21549 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
LMNA P02545 2/20 0.36
HPGD P15428 1/20 0.36
GAA P10253 1/20 0.36
GFER P55789 1/20 0.36
MPO P05164 1/20 0.36
SLC6A4 P31645 1/20 0.36
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28826421 0.73 IDO1 (0.38) ALDH1A1CYP2D6ATMIDO1AGXT
SCHEMBL9602890 0.67 ALDH1A1 (0.37) ALDH1A1CYP2D6ATMIDO1AGXT
SCHEMBL1172247 0.66 ALDH1A1 (0.41) ALDH1A1IDO1TAAR1LMNAGAA
SCHEMBL1824702 0.65 MAOB (0.55) ALDH1A1CYP2D6IDO1AGXTTAAR1
SCHEMBL1171878 0.65 ALDH1A1 (0.35) ALDH1A1HPGDGAAPOLB
Hydrochloric Acid SCHEMBL30293103 0.64 MAOB (0.53) ALDH1A1IDO1AGXTTAAR1SLC6A4
SCHEMBL9602886 0.64 LMNA (0.38) ALDH1A1CYP2D6ATMIDO1AGXT
SCHEMBL1822033 0.63 MAOB (0.47) IDO1AGXTTAAR1SLC6A4
SCHEMBL491284 0.63 IDO1 (0.42) ALDH1A1CYP2D6IDO1AGXTTAAR1
SCHEMBL4868046 0.62 TDP1 (0.52) ALDH1A1IDO1AGXTTAAR1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed