SCHEMBL28828433

SCHEMBL28828433

Cc1ccc(-c2ccc3c(c2)CC(C)(C)C3OC(N)=O)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.34
AKR1C2 P52895 2/20 0.34
AKR1B10 O60218 1/20 0.34
AKR1C4 P17516 1/20 0.34
AKR1C1 Q04828 1/20 0.34
KDM1A O60341 4/20 0.33
BACE1 P56817 1/20 0.33
GRM2 Q14416 1/20 0.33
JAK2 O60674 1/20 0.32
CTSA P10619 1/20 0.32
TDP2 O95551 1/20 0.31
OTUD7B Q6GQQ9 1/20 0.31
APP P05067 3/20 0.31
CYP3A4 P08684 3/20 0.31
CYP2C9 P11712 3/20 0.31
CYP2C19 P33261 3/20 0.31
CYP2D6 P10635 2/20 0.31
CYP1A2 P05177 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28828442 0.91 OTUD7B (0.39) BACE1CTSAOTUD7BAPPRORC
SCHEMBL28828624 0.90 TDP2 (0.41) BACE1GRM2TDP2APPCYP3A4
SCHEMBL28828429 0.88 KDM1A (0.33) KDM1ARORC
SCHEMBL29121265 0.87 AKR1C3 (0.38) AKR1C3AKR1C2KDM1AGRM2CTSA
SCHEMBL28828754 0.87 AKR1C3 (0.38) AKR1C3AKR1C2KDM1AGRM2CTSA
SCHEMBL28828681 0.87 ABL1 (0.38) BACE1APP
SCHEMBL28828631 0.87 ACMSD (0.37) JAK2HDAC1RORC
SCHEMBL28828584 0.86 APP (0.41) AKR1C3AKR1C2AKR1C1APPHDAC1
SCHEMBL28828434 0.86 MPL (0.33) HDAC1RORC
SCHEMBL28828382 0.85 DHODH (0.36) JAK2TDP2CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN claimed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN claimed
CN-114829361-B Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing the same 柳韩洋行 2024-07-16 CN disclosed
CN-114829361-A Derivatives having 2, 3-dihydro-1H-indene or 2, 3-dihydrobenzofuran moiety or pharmaceutically acceptable salts thereof and pharmaceutical compositions containing same 柳韩洋行 2022-07-29 CN disclosed