SCHEMBL28833973

SCHEMBL28833973

CC(C)(C)OC(=O)N1CC[C@H](Nc2cc(C(F)(F)F)cc3ncccc23)C1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.48
CNR1 P21554 3/20 0.46
USP30 Q70CQ3 5/20 0.46
PIK3CD O00329 1/20 0.46
MET P08581 1/20 0.44
TRPV1 Q8NER1 1/20 0.44
SYK P43405 1/20 0.44
BRD4 O60885 1/20 0.44
IDH1 O75874 1/20 0.44
BTK Q06187 1/20 0.43
STS P08842 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
PIK3CA P42336 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28833974 1.00 TACR1 (0.48) TACR1CNR1USP30PIK3CDMET
SCHEMBL29862929 1.00 TACR1 (0.48) TACR1CNR1USP30PIK3CDMET
SCHEMBL29862440 1.00 TACR1 (0.48) TACR1CNR1USP30PIK3CDMET
SCHEMBL28833985 1.00 TACR1 (0.48) TACR1CNR1USP30PIK3CDMET
SCHEMBL29863261 0.89 USP30 (0.47) CNR1USP30PIK3CDBRD4BTK
SCHEMBL28833993 0.89 USP30 (0.47) CNR1USP30PIK3CDBRD4BTK
SCHEMBL29862687 0.89 USP30 (0.47) CNR1USP30PIK3CDBRD4BTK
SCHEMBL28833994 0.89 USP30 (0.47) CNR1USP30PIK3CDBRD4BTK
SCHEMBL28834141 0.89 USP30 (0.47) CNR1USP30PIK3CDBRD4BTK
SCHEMBL23359881 0.87 CRHR1 (0.41) TACR1TRPV1SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055014-B1 PYRROLIDINE AND PIPERIDINE COMPOUNDS YUHAN CORP (KR) 2025-04-30 EP disclosed
CN-114867719-B Pyrrolidine and piperidine compounds 柳韩洋行 2024-06-25 CN disclosed
US-11655235-B2 Pyrrolidine and piperidine compounds YUHAN CORPORATION (KR) 2023-05-23 US disclosed
EP-4055014-A1 PYRROLIDINE AND PIPERIDINE COMPOUNDS Yuhan Corporation (KR) 2022-09-14 EP disclosed
CN-114867719-A Pyrrolidine and piperidine compounds 柳韩洋行 2022-08-05 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11655235-B2 Pyrrolidine and piperidine compounds FAP, APC, VHL TACR1 1681/4885CNR1 3970/4885USP30 1231/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.