SCHEMBL288348

SCHEMBL288348

Cc1ccc(-c2nccn2S(N)(=O)=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 6/20 0.39
CA9 Q16790 5/20 0.39
CA1 P00915 5/20 0.39
CA12 O43570 4/20 0.39
CA5A P35218 2/20 0.39
CA5B Q9Y2D0 2/20 0.39
CA3 P07451 1/20 0.39
CA6 P23280 1/20 0.39
CA7 P43166 1/20 0.39
RECQL P46063 1/20 0.39
PTGS2 P35354 6/20 0.39
TNKS O95271 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PTGS1 P23219 3/20 0.38
TSHR P16473 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL770698 0.77 L3MBTL1 (0.50) CA2CA1L3MBTL1TSHRMEN1
SCHEMBL28175124 0.75 POLB (0.45) CA2CA9CA1CA12RECQL
SCHEMBL1955893 0.75 CA1 (0.42) CA2CA9CA1CA12CA5A
SCHEMBL28303263 0.73 L3MBTL1 (0.54) CA2CA1L3MBTL1TSHRALDH1A1
SCHEMBL27556606 0.73 TNKS (0.41) TNKSMEN1KMT2AALDH1A1
SCHEMBL10194263 0.71 KDM4E (0.51) TNKSL3MBTL1TSHRMEN1KMT2A
SCHEMBL27549719 0.69 HPGD (0.40) TNKSMEN1KMT2AALDH1A1
SCHEMBL27826039 0.69 NISCH (0.38) TNKSMEN1KMT2AALDH1A1
SCHEMBL28008031 0.69 NISCH (0.38) TNKSMEN1KMT2AALDH1A1
SCHEMBL8636455 0.69 ESR1 (0.45) CA2CA9CA1CA12CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 76 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109923112-A Kill the oxadiazole derivatives of microorganism 先正达参股股份有限公司 2019-06-21 CN disclosed
CN-109890209-A Kill the oxadiazole derivatives of microorganism 先正达参股股份有限公司 2019-06-14 CN disclosed
CN-109071522-A Microbicidal oxadiazole derivatives 先正达参股股份有限公司 2018-12-21 CN disclosed
CN-108760920-A A method of cyazofamid and its metabolite residue amount are measured based on HPLC-MSMS methods 山东省农药科学研究院 2018-11-06 CN disclosed
EP-2922831-A1 PESTICIDAL COMPOUNDS BASED ON ARYLTHIOSULFONAMIDE DERIVATIVES Syngenta Participations AG (CH) 2015-09-30 EP disclosed
EP-2922837-A1 INSECTICIDAL COMPOUNDS BASED ON N-(ARYLSULFANYLMETHYL) CARBOXAMIDE DERIVATIVES Syngenta Participations AG (CH) 2015-09-30 EP disclosed
EP-2917201-A1 DIHYDROTHIOPHENE DERIVATIVES AS INSECTICIDAL COMPOUNDS Syngenta Participations AG (CH) 2015-09-16 EP disclosed
EP-2887810-A1 METHODS OF CONTROLLING INSECTS Syngenta Participations AG (CH) 2015-07-01 EP disclosed
EP-2887809-A1 METHODS OF CONTROLLING INSECTS Syngenta Participations AG (CH) 2015-07-01 EP disclosed
EP-2887802-A2 METHODS OF SOIL PEST CONTROL Syngenta Participations AG (CH) 2015-07-01 EP disclosed
WO-2011067135-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067240-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067131-A1 SPIROHETEROCYCLIC DIONE DERIVATIVES USED AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067203-A1 CHEMICAL COMPOUNDS AND THEIR USE AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067272-A1 INSECTICIDAL COMPOUNDS BASED ON ISOXAZOLINE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
EP-2324010-A1 INSECTICIDAL PHENYL- OR PYRIDYL-PIPERIDINE COMPOUNDS Syngenta Participations AG (CH) 2011-05-25 EP disclosed
WO-2011003684-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2011-01-13 WO disclosed
WO-2010066780-A1 SPIROHETEROCYCLIC N-OXYPIPERIDINES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-06-17 WO disclosed
WO-2010063670-A1 SPIROHETEROCYCLIC N-OXYAMIDES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-06-10 WO disclosed
WO-2001055140-A1 ISOTHIAZOLE DERIVATIVES AND THEIR USE AS PESTICIDES SYNGENTA LIMITED (GB) 2001-08-02 WO disclosed