SCHEMBL288353

SCHEMBL288353

CN1CC(C(=O)O)NC1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.40
HTT P42858 1/20 0.39
CYP2D6 P10635 2/20 0.37
LMNA P02545 2/20 0.37
BLM P54132 2/20 0.37
ALOX15 P16050 2/20 0.37
CYP1A2 P05177 2/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
RAB9A P51151 1/20 0.37
MEN1 O00255 1/20 0.37
THRB P10828 1/20 0.37
PMP22 Q01453 1/20 0.37
KMT2A Q03164 1/20 0.37
IDUA P35475 1/20 0.36
CAD P27708 2/20 0.35
ACE P12821 1/20 0.35
GRM2 Q14416 1/20 0.34
GRM3 Q14832 1/20 0.34
EGLN1 Q9GZT9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6999553 1.00 P2RX7 (0.40) P2RX7HTTCYP2D6LMNABLM
SCHEMBL5081569 1.00 P2RX7 (0.40) P2RX7HTTCYP2D6LMNABLM
SCHEMBL5365854 1.00 P2RX7 (0.40) P2RX7HTTCYP2D6LMNABLM
Hydrochloric Acid SCHEMBL28572830 0.98 P2RX7 (0.39) P2RX7HTTCYP2D6LMNABLM
SCHEMBL8232195 0.83 P2RX7 (0.40) P2RX7
SCHEMBL25251069 0.81 P2RX7 (0.39) P2RX7ACE
SCHEMBL8067332 0.81 P2RX7 (0.36) P2RX7
Lithium Ion SCHEMBL30619228 0.79 P2RX7 (0.38) P2RX7
SCHEMBL6992243 0.79 HTT (0.37) HTTCYP2D6LMNABLMALOX15
SCHEMBL8231725 0.78 BRD4 (0.49) P2RX7CYP1A2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 75 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007029267-A1 PROCESS FOR INDUSTRIALLY VIABLE PREPARATION OF IMIDAPRIL HYDROCHLORIDE POTLURI RAMESH BABU (IN) 2007-03-15 WO claimed
EP-3985001-B1 PHARMACEUTICAL COMPOSITION FOR USE IN TREATING A CANCER SERVIER LAB (FR) 2026-04-29 EP disclosed
EP-4631573-A2 TEAD INHIBITORS Orion Corporation (FI) 2025-10-15 EP disclosed
EP-4323338-B1 TEAD INHIBITORS ORION CORP (FI) 2025-10-08 EP disclosed
US-20240158392-A1 SMALL MOLECULE INHIBITORS OF SALT INDUCIBLE KINASES JANSSEN RESEARCH & DEVELOPMENT, LLC 2024-05-16 US disclosed
US-20240059733-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE SERVIER PHARMACEUTICALS LLC (US) 2024-02-22 US disclosed
EP-4284801-A1 SMALL MOLECULE INHIBITORS OF SALT INDUCIBLE KINASES Janssen Biotech, Inc. (US) 2023-12-06 EP disclosed
WO-2023205618-A2 CCR4 ANTAGONISTS CHEMOCENTRYX, INC. (US) 2023-10-26 WO disclosed
US-11667673-B2 Therapeutically active compounds and their methods of use SERVIER PHARMACEUTICALS LLC (US) 2023-06-06 US disclosed
EP-3985001-A1 PHARMACEUTICAL COMPOSITION USEFUL IN INHIBITING IDH1 Les Laboratoires Servier SAS (FR) 2022-04-20 EP disclosed
CN-1139599-C Process for the preparation of pharmacologically acceptable salts of N- (1(S) -ethoxycarbonyl-3-phenylpropyl) -L-alanyl-amino acids ��Ԩ��ѧ��ҵ��ʽ���� 2004-02-25 CN disclosed
US-20030105327-A1 Process for preparing pharmacologically acceptable salt of N-(1(S)-ethoxycarbonyl-3-phenylpropyl)-L-alanyl-amino acid KANEKA CORPORATION (JP) 2003-06-05 US disclosed
US-6518436-B2 Condensing an amino acid and N-(1(S)-ethoxycarbonyl-3-phenylpropyl)-L-alanine-N-carboxy-anhydride; suppressing the by-product diketopiperazine derivative; making enalapril maleate KANEKA CORPORATION (JP) 2003-02-11 US disclosed
US-20020087007-A1 Process for preparing pharmacologically acceptable salt of N-(1(S)-ethoxycarbonyl-3-phenylpropyl)-L-alanyl-amino acid KANEKA CORPORATION (JP) 2002-07-04 US disclosed
US-6335453-B1 BY-PROUDCT INHIBITION KANEKA CORPORATION (JP) 2002-01-01 US disclosed
EP-0967221-A1 PROCESS FOR PREPARING PHARMACOLOGICALLY ACCEPTABLE SALTS OF N-(1(S)-ETHOXYCARBONYL-3-PHENYLPROPYL)-L-ALANYL AMINO ACIDS KANEKA CORPORATION (JP) 1999-12-29 EP disclosed
CN-1234804-A Process for preparing pharmacologically acceptable salts of N-(1-(S)-ethoxycarbonyl-3-phenylpropyl)-L-alanyl amino acids KANEKA CHEMICAL IND CO LTD (JP) 1999-11-10 CN disclosed
EP-0373881-A2 Process for preparing optically active 2-oxoimidazolidine derivatives TANABE SEIYAKU CO., LTD. (JP) 1990-06-20 EP disclosed
EP-0095163-A2 2-Oxo-imidazolidine compounds, a process for preparing the same and a pharmaceutical composition Tanabe Seiyaku Co., Ltd. (JP) 1983-11-30 EP disclosed
EP-0052696-A1 Novel 2-oxoimidazolidine derivative, a process for preparing same and a pharmaceutical composition containing the 2-oxoimidazolidine derivative Tanabe Seiyaku Co., Ltd. (JP) 1982-06-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240158392-A1 SMALL MOLECULE INHIBITORS OF SALT INDUCIBLE KINASES SIK2, SIK1, SGK2 P2RX7 4769/4885HTT 3602/4885CYP2D6 4759/4885
US-20030105327-A1 Process for preparing pharmacologically acceptable salt of N-(1(S)-ethoxycarbonyl-3-phenylpropyl)-L-alanyl-amino acid SLC7A1, ASS1, ALDH7A1 P2RX7 3949/4885HTT 1738/4885CYP2D6 1307/4885
US-20240059733-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE IDH1, IDH3B, IDH3A P2RX7 4549/4885HTT 303/4885CYP2D6 1949/4885
US-20020087007-A1 Process for preparing pharmacologically acceptable salt of N-(1(S)-ethoxycarbonyl-3-phenylpropyl)-L-alanyl-amino acid SLC7A1, ASS1, ALDH7A1 P2RX7 3949/4885HTT 1738/4885CYP2D6 1307/4885
US-11667673-B2 Therapeutically active compounds and their methods of use IDH1, IDH3B, IDH3A P2RX7 4549/4885HTT 303/4885CYP2D6 1949/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.