SCHEMBL28836368

SCHEMBL28836368

COC(=O)Cc1cn(C)c2cc(F)ccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
IDO1 P14902 1/20 0.46
TDO2 P48775 1/20 0.46
CDK2 P24941 1/20 0.46
KDM4E B2RXH2 2/20 0.44
MAPT P10636 4/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.42
TSHR P16473 1/20 0.42
S1PR2 O95136 1/20 0.41
LMNA P02545 2/20 0.40
TP53 P04637 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
AKR1C3 P42330 1/20 0.40
DRD2 P14416 1/20 0.40
SLC6A4 P31645 1/20 0.40
ICMT O60725 2/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14564357 0.84 ICMT (0.47) MEN1KMT2ACDK2KDM4EMAPT
SCHEMBL2085331 0.84 KDM4E (0.51) MEN1KMT2AKDM4EMAPTALDH1A1
SCHEMBL30275134 0.84 MEN1 (0.50) MEN1KMT2AIDO1TDO2CDK2
SCHEMBL5447791 0.83 KDM4E (0.44) MEN1KMT2AKDM4EMAPTALDH1A1
SCHEMBL31498840 0.80 KDM4E (0.65) MEN1KMT2AKDM4EMAPTALDH1A1
SCHEMBL4012453 0.80 KDM4E (0.65) MEN1KMT2AKDM4EMAPTALDH1A1
SCHEMBL18508627 0.79 DRD2 (0.50) MEN1KMT2AIDO1TDO2CDK2
SCHEMBL7524516 0.78 MAPT (0.44) MEN1KMT2AKDM4EMAPTALDH1A1
SCHEMBL2081872 0.78 ALDH1A1 (0.40) MEN1KMT2AKDM4EMAPTALDH1A1
SCHEMBL30275080 0.77 LMNA (0.48) MEN1KMT2AIDO1TDO2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113292557-B Pyridopyrimidinone mesoion derivative containing indole unit and preparation method and application thereof 贵州大学 2022-02-11 CN disclosed
CN-113292557-A Pyridopyrimidinone mesoion derivative containing indole unit and preparation method and application thereof 贵州大学 2021-08-24 CN disclosed