SCHEMBL28837181

SCHEMBL28837181

N#Cc1cncnc1-c1ccccc1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.43
ADORA1 P30542 1/20 0.43
SLC22A12 Q96S37 2/20 0.40
ALDH1A1 P00352 4/20 0.38
CYP1A2 P05177 3/20 0.38
CYP3A4 P08684 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
MEN1 O00255 1/20 0.38
THRB P10828 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
IDO1 P14902 2/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
PDK1 Q15118 1/20 0.36
HSD17B10 Q99714 2/20 0.36
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
ATR Q13535 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27848361 0.79 CNR1 (0.38) SLC22A12ALDH1A1CYP3A4TDP1CNR1
SCHEMBL10460219 0.77 SLC22A12 (0.45) ADORA2AADORA1SLC22A12ALDH1A1CYP1A2
SCHEMBL25417900 0.76 ADORA2A (0.56) ADORA2AADORA1SLC22A12ALDH1A1TDP1
SCHEMBL29974619 0.72 EPHB3 (0.41) SLC22A12GABRA1GABRG2GABRB3GABRA3
SCHEMBL30219258 0.70 IMPDH2 (0.54) ALDH1A1CYP1A2CYP3A4MEN1HPGD
SCHEMBL12006859 0.69 ALDH1A1 (0.59) ALDH1A1CYP1A2CYP3A4MEN1HPGD
SCHEMBL166305 0.69
SCHEMBL30747854 0.69 MAPK9 (0.57) ADORA2AADORA1ALDH1A1THRBPDK1
SCHEMBL17144583 0.67 LRRK2 (0.58)
SCHEMBL2652308 0.67 GABRG2 (0.47) SLC22A12PDK1GABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106170290-A Substituted di-amino-pyrimidine based compound, combinations thereof and treatment method thereof 西格诺药品有限公司 2016-11-30 CN disclosed