SCHEMBL2884296

SCHEMBL2884296

Nc1ccc(-c2ccc(F)cc2F)nc1N

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
ADORA2A P29274 2/20 0.48
ADORA1 P30542 2/20 0.48
KMO O15229 2/20 0.45
HDAC1 Q13547 8/20 0.41
HDAC2 Q92769 8/20 0.41
ALPL P05186 2/20 0.40
KIT P10721 1/20 0.37
F2RL3 Q96RI0 1/20 0.37
MPL P40238 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL898443 0.86 ALDH1A1 (0.45) ALDH1A1ADORA2AADORA1MPL
SCHEMBL20738436 0.83 ALDH1A1 (0.47) ALDH1A1ADORA2AADORA1KMOHDAC1
SCHEMBL21811276 0.79 KMO (0.57) ALDH1A1ADORA2AADORA1KMOHDAC1
SCHEMBL1582795 0.78 MPL (0.53) ALDH1A1ADORA2AMPL
SCHEMBL11906681 0.78 KMO (0.56) ALDH1A1ADORA2AADORA1KMOHDAC1
SCHEMBL9887058 0.77 TDP1 (0.54) ALDH1A1ADORA2AADORA1KMOHDAC1
SCHEMBL23190261 0.76 HDAC1 (0.47) ALDH1A1ADORA2AADORA1KMOHDAC1
SCHEMBL3923995 0.75 KMO (0.45) ALDH1A1ADORA2AADORA1KMOALPL
SCHEMBL13261826 0.75 KMO (0.51) ADORA2AADORA1KMOALPLF2RL3
SCHEMBL21811205 0.74 ALPL (0.54) KMOHDAC1HDAC2ALPLF2RL3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021016413-A1 SYNTHESIS OF BICYCLIC INHIBITORS OF HISTONE DEACETYLASE ALKERMES, INC. (US) 2021-01-28 WO disclosed
US-7691860-B2 Sulfonamide derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 2010-04-06 US disclosed
US-20080161326-A1 Novel Sulfone Amide Amide Derivatives MSD K.K. (JP) 2008-07-03 US disclosed
EP-1719765-A1 NOVEL SULFONE AMIDE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2006-11-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080161326-A1 Novel Sulfone Amide Amide Derivatives NPY1R, NPY2R, NPY5R ALDH1A1 1680/4885ADORA2A 1506/4885ADORA1 899/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.