SCHEMBL28845072

SCHEMBL28845072

Fc1cccc(-c2cccnn2)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.41
CASP6 P55212 1/20 0.39
HSD11B1 P28845 1/20 0.36
HTR2C P28335 3/20 0.36
HDAC4 P56524 1/20 0.36
GABRG2 P18507 4/20 0.35
GABRB3 P28472 4/20 0.35
GABRA5 P31644 4/20 0.35
GABRA3 P34903 4/20 0.35
BCAT1 P54687 1/20 0.35
NPY5R Q15761 1/20 0.35
GABRA1 P14867 2/20 0.35
NOTUM Q6P988 1/20 0.34
HTR2A P28223 2/20 0.34
CDK2 P24941 2/20 0.34
CCNE2 O96020 1/20 0.34
CCNE1 P24864 1/20 0.34
HTR2B P41595 1/20 0.33
WDR5 P61964 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25180819 0.85 CASP6 (0.36) FAAHCASP6HTR2CHDAC4GABRG2
SCHEMBL28211033 0.84 GABRG2 (0.47) CASP6HDAC4GABRG2GABRB3GABRA5
SCHEMBL34461976 0.84 GABRG2 (0.47) CASP6HDAC4GABRG2GABRB3GABRA5
SCHEMBL23499270 0.78 CASP6 (0.40) FAAHCASP6HTR2CHDAC4GABRG2
SCHEMBL16711570 0.78 GABRG2 (0.43) CASP6HTR2CHDAC4GABRG2GABRB3
SCHEMBL1248582 0.77 FAAH (0.33) FAAH
SCHEMBL30888806 0.74 KDM4E (0.50) MAPK1
SCHEMBL970044 0.74 KDM4E (0.50) MAPK1
SCHEMBL24352491 0.74 CASP6 (0.41) CASP6HTR2CHDAC4GABRG2GABRB3
SCHEMBL29986122 0.73 KDM4E (0.48) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103002897-B Certain amino-pyridazines, compositions thereof, and methods of use thereof 赛特凯恩蒂克公司 2017-06-09 CN claimed