SCHEMBL2884549

SCHEMBL2884549

Nc1ccc(Cl)c(Oc2cc(Cl)cc(Br)c2Cl)c1[N+](=O)[O-]

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
TSHR P16473 2/20 0.37
PDE7A Q13946 2/20 0.35
EPAS1 Q99814 2/20 0.33
VEGFA P15692 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HTT P42858 2/20 0.32
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
XBP1 P17861 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TLR9 Q9NR96 1/20 0.32
THRA P10827 2/20 0.32
TDP1 Q9NUW8 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL4440818 0.93 ALDH1A1 (0.33) ALDH1A1TSHRPDE7AEPAS1VEGFA
SCHEMBL2880917 0.80 TSHR (0.32) TSHRTP53CYP3A4
SCHEMBL2943368 0.79 MEN1 (0.38) ALDH1A1TSHRPDE7AEPAS1VEGFA
SCHEMBL2878659 0.77 ALDH1A1 (0.47) ALDH1A1TSHRPDE7AMEN1KMT2A
Iodide SCHEMBL4440824 0.77 ALDH1A1 (0.31) ALDH1A1TSHREPAS1VEGFA
SCHEMBL4786052 0.75 MEN1 (0.36) ALDH1A1TSHRPDE7AEPAS1VEGFA
SCHEMBL22326087 0.69 PDE7A (0.42) ALDH1A1PDE7AMEN1KMT2AHTT
SCHEMBL22325952 0.68 EPAS1 (0.46) ALDH1A1PDE7AEPAS1MEN1KMT2A
SCHEMBL31330060 0.68 ALDH1A1 (0.42) ALDH1A1TSHRPDE7AMEN1KMT2A
SCHEMBL240637 0.68 PTGER4 (0.48) ALDH1A1TSHRMEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121638-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS MERCK SHARP & DOHME (US) 2016-05-25 EP disclosed
US-20100286192-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS ANTHONY NEVILLE J 2010-11-11 US disclosed
US-7781454-B2 Non-nucleoside reverse transcriptase inhibitors MERCK SHARP & DOHME CORP. (US) 2010-08-24 US disclosed
EP-2121638-A2 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS Merck & Co., Inc. (US) 2009-11-25 EP disclosed
US-20080275097-A1 Non-nucleoside reverse transcriptase inhibitors MERCK SHARP & DOHME LLC 2008-11-06 US disclosed
WO-2008076225-A2 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS MERCK & CO., INC. (US) 2008-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080275097-A1 Non-nucleoside reverse transcriptase inhibitors RNGTT, RRM2B, RRM2 ALDH1A1 2863/4885TSHR 2632/4885PDE7A 1715/4885
US-20100286192-A1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS RNGTT, RRM2B, RRM2 ALDH1A1 2863/4885TSHR 2632/4885PDE7A 1715/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.