SCHEMBL28845803

SCHEMBL28845803

Nc1cnc(-c2cc([N+](=O)[O-])ccc2F)nc1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 5/20 0.44
ALDH1A1 P00352 4/20 0.43
HIF1A Q16665 1/20 0.43
AMY1A P0DUB6 1/20 0.40
CYP3A4 P08684 4/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
TSHR P16473 2/20 0.39
GAA P10253 1/20 0.39
THRB P10828 1/20 0.39
TLR2 O60603 2/20 0.38
TLR1 Q15399 2/20 0.38
HSPB1 P04792 1/20 0.38
PTPRC P08575 1/20 0.37
S100A4 P26447 1/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MCL1 Q07820 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1582458 0.78 NPC1 (0.39) ALDH1A1
SCHEMBL29890962 0.75 WDR5 (0.48) ALDH1A1CYP3A4KMT2ACYP1A2CYP2C19
SCHEMBL28845844 0.75 WDR5 (0.48) ALDH1A1CYP3A4MEN1KMT2ACYP1A2
SCHEMBL28845825 0.75 WDR5 (0.48) ALDH1A1CYP3A4KMT2ACYP1A2CYP2C19
SCHEMBL6221321 0.75 ALDH1A1 (0.51) TDP1ALDH1A1HIF1AAMY1ACYP3A4
SCHEMBL4910527 0.74 ALDH1A1 (0.67) TDP1ALDH1A1HIF1AAMY1ACYP3A4
SCHEMBL2884342 0.71 DPP4 (0.43) ALDH1A1KDM4EHTT
SCHEMBL27612318 0.71 TDP1 (0.48) TDP1ALDH1A1HIF1AAMY1ACYP3A4
SCHEMBL18495641 0.71 CLK1 (0.60) TDP1ALDH1A1HIF1AAMY1AMAPT
SCHEMBL589324 0.70 ALDH1A1 (0.62) TDP1ALDH1A1HIF1ACYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109734674-B Aniline WDR5 protein-protein interaction inhibitor and preparation method and application thereof 中国药科大学 2022-08-26 CN disclosed