SCHEMBL28849065

SCHEMBL28849065

COC(=O)c1cccc(C2(C(F)(F)F)CC2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 3/20 0.49
RAB9A P51151 3/20 0.46
POLB P06746 1/20 0.46
ALDH1A1 P00352 2/20 0.44
LOXL2 Q9Y4K0 1/20 0.44
MRGPRX4 Q96LA9 1/20 0.44
NPC1 O15118 2/20 0.43
TSHR P16473 1/20 0.43
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
SDHB P21912 1/20 0.43
MDH1 P40925 1/20 0.42
MDH2 P40926 1/20 0.42
MAPT P10636 2/20 0.42
HPGD P15428 1/20 0.42
EPHX2 P34913 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
NOTUM Q6P988 1/20 0.42
TP53 P04637 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21036244 0.81 CA1 (0.47) PDK2RAB9APOLBALDH1A1LOXL2
SCHEMBL28168249 0.81 KDM4C (0.46) PDK2ALDH1A1HPGD
SCHEMBL12985400 0.79 PDK2 (0.46) PDK2RAB9APOLBALDH1A1LOXL2
SCHEMBL24852732 0.79 NOTUM (0.40) PDK2RAB9APOLBALDH1A1NPC1
SCHEMBL29918286 0.79 NOTUM (0.40) PDK2RAB9APOLBALDH1A1NPC1
SCHEMBL3942652 0.78 LOXL2 (0.49) RAB9APOLBALDH1A1LOXL2NPC1
SCHEMBL21609774 0.78 NOTUM (0.56) PDK2POLBNOTUM
SCHEMBL17709905 0.78 NOTUM (0.56) PDK2POLBALDH1A1MAPTEPHX2
SCHEMBL21296558 0.77 SIGMAR1 (0.37) ALDH1A1TSHRMAPTEPHX2OPRM1
SCHEMBL1670244 0.77 LOXL2 (0.51) RAB9APOLBALDH1A1LOXL2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107108598-A Thiazoles as Ror gamma t modulators 詹森药业有限公司 2017-08-29 CN disclosed