SCHEMBL2884932

SCHEMBL2884932

O=Cc1cnc(C(=NOC2CC2)c2ccc(F)c(F)c2)nc1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.36
KCNQ3 O43525 4/20 0.34
KCNQ2 O43526 4/20 0.34
PLA2G7 Q13093 1/20 0.34
HSD11B1 P28845 1/20 0.34
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
NTSR1 P30989 1/20 0.32
KCNH2 Q12809 2/20 0.31
MCHR1 Q99705 2/20 0.31
RAB9A P51151 1/20 0.31
KCNQ5 Q9NR82 1/20 0.31
CHRNA7 P36544 1/20 0.31
SSTR3 P32745 2/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
VNN1 O95497 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2884930 1.00 AR (0.36) ARKCNQ3KCNQ2PLA2G7HSD11B1
SCHEMBL2882433 0.81 AR (0.32) ARKCNQ3KCNQ2HSD11B1CES2
SCHEMBL4066477 0.73 CES2 (0.46) KCNQ3KCNQ2PLA2G7CES2CES1
SCHEMBL2880794 0.73 MCHR1 (0.40) KCNH2MCHR1
SCHEMBL4068874 0.61 CES2 (0.44) KCNQ3KCNQ2PLA2G7CES2CES1
SCHEMBL28004400 0.60 SERPINE1 (0.56) KCNQ3KCNQ2PLA2G7HSD11B1CES2
SCHEMBL28266834 0.58 SERPINE1 (0.51) PLA2G7HSD11B1CES2CES1RAB9A
SCHEMBL21448795 0.58 HSD11B1 (0.60) HSD11B1CES2CES1RAB9AMEN1
Ethylene Glycol SCHEMBL28725409 0.56 ALDH1A1 (0.44) PLA2G7CES2CES1RAB9A
SCHEMBL48607 0.56 ALDH1A1 (0.52) PLA2G7CES2CES1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100324049-A1 DIARYL KETIMINE DERIVATIVE HAVING ANTAGONISM AGAINST MELANIN-CONCENTRATING HORMONE RECEPTOR MSD K.K. (JP) 2010-12-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100324049-A1 DIARYL KETIMINE DERIVATIVE HAVING ANTAGONISM AGAINST MELANIN-CONCENTRATING HORMONE RECEPTOR MC1R, MCHR1, MCHR2 AR 47/4885KCNQ3 987/4885KCNQ2 1125/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.