SCHEMBL28853404

SCHEMBL28853404

COC(=O)c1ccccc1Oc1cc(C(F)(F)F)nc(C)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
SDHB P21912 1/20 0.50
ALDH1A1 P00352 3/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
KDM4E B2RXH2 3/20 0.43
POLB P06746 1/20 0.43
TP53 P04637 1/20 0.42
CYP1A2 P05177 3/20 0.41
CYP2C9 P11712 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP3A4 P08684 2/20 0.41
MAPK1 P28482 1/20 0.41
MAPK8 P45983 1/20 0.41
MAPK10 P53779 1/20 0.41
SLC6A3 Q01959 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
HPGD P15428 1/20 0.41
ATM Q13315 1/20 0.41
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29113152 0.80 TUBB4A (0.43) SDHBALDH1A1KDM4EPOLBCYP1A2
SCHEMBL17623925 0.78 HTT (0.46) MEN1KMT2AALDH1A1KDM4EPOLB
SCHEMBL30636497 0.78 ALDH1A1 (0.56) SDHBALDH1A1SMN1; SMN2KDM4EPOLB
SCHEMBL28853408 0.78 ALDH1A1 (0.56) SDHBALDH1A1SMN1; SMN2KDM4EPOLB
SCHEMBL17623924 0.73 BLM (0.58) MEN1KMT2ASDHBALDH1A1KDM4E
SCHEMBL16302025 0.72 SCN8A (0.53) TDP1
SCHEMBL2441955 0.72 SLC6A3 (0.65) MEN1KMT2AALDH1A1SMN1; SMN2KDM4E
SCHEMBL10338670 0.71 KMT2A (0.73) MEN1KMT2AALDH1A1SMN1; SMN2KDM4E
SCHEMBL4318924 0.71 ALDH1A1 (0.69) MEN1KMT2AALDH1A1SMN1; SMN2KDM4E
SCHEMBL9024615 0.71 BDKRB1 (0.52) SDHBSLC6A3SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115124475-A Pyrimidine derivative and preparation method and application thereof 贵阳学院 2022-09-30 CN claimed
CN-115124475-A Pyrimidine derivative and preparation method and application thereof 贵阳学院 2022-09-30 CN disclosed