SCHEMBL28854243

SCHEMBL28854243

C[C@H](NC(=O)OC(C)(C)C)c1cn[nH]c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.47
TSHR P16473 3/20 0.46
HSD17B10 Q99714 2/20 0.46
ALDH1A1 P00352 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TRPA1 O75762 1/20 0.40
MAPT P10636 1/20 0.40
ATM Q13315 1/20 0.40
CTSK P43235 2/20 0.40
CYP2C8 P10632 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38
ACACB O00763 1/20 0.38
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28854244 1.00 KMT2A (0.47) KMT2ATSHRHSD17B10ALDH1A1L3MBTL1
SCHEMBL32681721 0.82 CTSS (0.43) KMT2ATRPA1ATMCTSKCA1
SCHEMBL18869910 0.80 ROCK2 (0.53)
SCHEMBL15336444 0.80 ROCK2 (0.53)
SCHEMBL28200955 0.76 CTSK (0.43) KMT2ATSHRHSD17B10TRPA1MAPT
SCHEMBL28200954 0.76 CTSK (0.43) KMT2ATSHRHSD17B10TRPA1MAPT
SCHEMBL21208148 0.75 STK17B (0.40) KMT2AALDH1A1CA1CA2LMNA
SCHEMBL6947166 0.75 CTSK (0.47) KMT2ATSHRHSD17B10ALDH1A1L3MBTL1
SCHEMBL14127863 0.75 KMT2A (0.43) KMT2ATSHRHSD17B10ALDH1A1L3MBTL1
SCHEMBL12203593 0.74 CTSK (0.62) KMT2AHSD17B10ALDH1A1MAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107474050-A 6,7 dihydro-pyrazolos [1,5 a] pyrazine 4 (5H) assimilation compound 詹森药业有限公司 2017-12-15 CN disclosed