SCHEMBL28859253

SCHEMBL28859253

C#Cc1ccccc1N(CC=C)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.36
GSTO1 P78417 1/20 0.36
TSHR P16473 1/20 0.36
BCL2A1 Q16548 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 3/20 0.32
MAPT P10636 2/20 0.32
HPGD P15428 2/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
THRB P10828 1/20 0.32
HIF1A Q16665 1/20 0.32
RAB9A P51151 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
C5AR1 P21730 1/20 0.31
POLB P06746 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28038900 0.82 CYP3A4 (0.43) L3MBTL1GSTO1TSHRNPSR1ALDH1A1
SCHEMBL23217979 0.81 ALDH1A1 (0.40) L3MBTL1GSTO1TSHRNPSR1KDM4E
SCHEMBL29009658 0.81 L3MBTL1 (0.38) L3MBTL1GSTO1TSHRBCL2A1NPSR1
SCHEMBL29096379 0.78 STAT5B (0.39) BCL2A1MEN1KMT2A
SCHEMBL6207086 0.77 L3MBTL1 (0.33) L3MBTL1GSTO1TSHRNPSR1KDM4E
SCHEMBL3221801 0.74 POLB (0.40) L3MBTL1GSTO1TSHRKDM4EALDH1A1
SCHEMBL15466723 0.74 SSTR4 (0.35) L3MBTL1GSTO1TSHRNPSR1KDM4E
SCHEMBL6205322 0.73 TSHR (0.34) L3MBTL1GSTO1TSHR
SCHEMBL20297003 0.73 L3MBTL1 (0.35) L3MBTL1GSTO1TSHRNPSR1KDM4E
SCHEMBL6207594 0.73 L3MBTL1 (0.33) L3MBTL1TSHRNPSR1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115043788-A Trifluoromethyl oxazole-2-ketone compound and preparation method and application thereof 南京工业大学 2022-09-13 CN claimed
CN-115043788-B Trifluoromethyl oxazol-2-one compound and preparation method and application thereof 南京工业大学 2023-10-20 CN disclosed