SCHEMBL28866622

SCHEMBL28866622

O=C(C(Br)c1ccsc1)C(Br)c1ccsc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.44
CES2 O00748 2/20 0.41
CES1 P23141 2/20 0.41
LCK P06239 1/20 0.40
FYN P06241 1/20 0.40
DAO P14920 1/20 0.40
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
HDAC1 Q13547 1/20 0.36
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KCNH2 Q12809 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7473459 0.85 CES2 (0.43) ALOX5CES2CES1LCKFYN
SCHEMBL7466610 0.83 ALOX5 (0.50) ALOX5CES2CES1LCKFYN
SCHEMBL5129994 0.79 ALOX5 (0.42) ALOX5CES2CES1LCKFYN
SCHEMBL27586694 0.78 ALOX5 (0.41) ALOX5CES2CES1LCKFYN
SCHEMBL28647770 0.76 ALOX5 (0.40) ALOX5CES2CES1LCKFYN
SCHEMBL4013434 0.76 CHRNB2 (0.43) ALOX5CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL27757242 0.75
SCHEMBL8716724 0.74 ALOX5 (0.53) ALOX5CES2CES1LCKFYN
SCHEMBL7827555 0.74
SCHEMBL27734035 0.74 ALOX5 (0.41) ALOX5CES2CES1LCKFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884103-A Tricyclic compounds as immunomodulators 正大天晴药业集团股份有限公司 2018-11-23 CN disclosed