SCHEMBL7473459

SCHEMBL7473459

O=C(O)C(Br)c1ccsc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.43
CES1 P23141 2/20 0.43
LCK P06239 1/20 0.43
FYN P06241 1/20 0.43
DAO P14920 1/20 0.43
ALOX5 P09917 1/20 0.43
IDO1 P14902 1/20 0.42
TDO2 P48775 1/20 0.42
HPGD P15428 1/20 0.38
SRC P12931 2/20 0.37
CYP2D6 P10635 1/20 0.37
SLC1A3 P43003 2/20 0.37
SLC1A2 P43004 2/20 0.37
SLC1A1 P43005 2/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
LMNA P02545 2/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28866622 0.85 ALOX5 (0.44) CES2CES1LCKFYNDAO
SCHEMBL7466610 0.82 ALOX5 (0.50) CES2CES1LCKFYNDAO
SCHEMBL28647770 0.79 ALOX5 (0.40) CES2CES1LCKFYNDAO
SCHEMBL162736 0.78 SRC (0.50) CES2CES1LCKFYNDAO
SCHEMBL18734632 0.78 CYP2D6 (0.50) CES2CES1LCKFYNDAO
SCHEMBL9462827 0.78 IDO1 (0.50) CES2CES1LCKFYNDAO
SCHEMBL5129994 0.77 ALOX5 (0.42) CES2CES1LCKFYNDAO
SCHEMBL9329422 0.77 LMNA (0.52) CES2CES1LCKFYNDAO
SCHEMBL200194 0.77 LMNA (0.52) CES2CES1LCKFYNDAO
Hydrochloric Acid SCHEMBL11244144 0.77 SRC (0.48) CES2CES1LCKFYNDAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077701-A4 ANTI-VIRAL COMPOUNDS LILLY CO ELI (US) 2002-03-20 EP disclosed
US-6358971-B1 FOR INHIBITING THE GROWTH OF A PICORNAVIRUS ELI LILLY AND COMPANY 2002-03-19 US disclosed
CN-1292697-A Anti-viral compound LILLY CO ELI (US) 2001-04-25 CN disclosed
EP-1077701-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 2001-02-28 EP disclosed
WO-1999059587-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 1999-11-25 WO disclosed
US-5843947-A N-pyridyl carboxamides and derivatives ADIR ET COMPAGNIE (FR) 1998-12-01 US disclosed
US-5712294-A N-pyridyl carboxamides and derivatives ADIR ET COMPAGNIE (FR) 1998-01-27 US disclosed
US-4329363-A Substituted mercapto acid amides and their use MERCK & CO., INC. (US) 1982-05-11 US disclosed
US-4216160-A IMMUNOREGULANTS FOR CORRECTING AN INBALANCE OF IMMUNE HOMEOSTASIS MERCK & CO., INC. (US) 1980-08-05 US disclosed
EP-0001989-A1 Substituted mercapto acid amides, process for their preparation, pharmaceutical composition containing same and their use MERCK & CO. INC. (US) 1979-05-30 EP disclosed
US-4110535-A BACTERICIDE E. R. SQUIBB & SONS, INC. (US) 1978-08-29 US disclosed
US-4088816-A BACTERICIDES E. R. SQUIBB & SONS, INC. (US) 1978-05-09 US disclosed
US-4052554-A BACTERICIDE E. R. SQUIBB & SONS, INC. (US) 1977-10-04 US disclosed
US-3996217-A BACTERICIDES E. R. SQUIBB & SONS, INC. (US) 1976-12-07 US disclosed
US-3996218-A BACTERICIDES E. R. SQUIBB & SONS, INC. (US) 1976-12-07 US disclosed